Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha

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Furans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0960-894X(01)00488-7
P698PubMed publication ID11549460

P2093author name stringSun J
Katzenellenbogen BS
Katzenellenbogen JA
Rodriguez AL
Mortensen DS
P2860cites workMolecular basis of agonism and antagonism in the oestrogen receptorQ27746278
The structural basis of estrogen receptor/coactivator recognition and the antagonism of this interaction by tamoxifenQ27766417
Estrogen receptor subtype-selective ligands: asymmetric synthesis and biological evaluation of cis- and trans-5,11-dialkyl- 5,6,11, 12-tetrahydrochrysenesQ28368417
Triarylpyrazoles with basic side chains: development of pyrazole-based estrogen receptor antagonistsQ31988135
The estradiol pharmacophore: ligand structure-estrogen receptor binding affinity relationships and a model for the receptor binding siteQ34419702
Novel ligands that function as selective estrogens or antiestrogens for estrogen receptor-alpha or estrogen receptor-betaQ34490307
Pyrazole ligands: structure-affinity/activity relationships and estrogen receptor-alpha-selective agonists.Q43517366
Synthesis and biological evaluation of a novel series of furans: ligands selective for estrogen receptor alphaQ43786351
Differential response of estrogen receptor alpha and estrogen receptor beta to partial estrogen agonists/antagonistsQ47866745
Regioselective synthesis of 1,3,5-triaryl-4-alkylpyrazoles: novel ligands for the estrogen receptorQ74240190
P433issue18
P407language of work or nameEnglishQ1860
P304page(s)2521-2524
P577publication date2001-09-01
P1433published inBioorganic & Medicinal Chemistry LettersQ2709483
P1476titleFurans with basic side chains: synthesis and biological evaluation of a novel series of antagonists with selectivity for the estrogen receptor alpha
P478volume11

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