Inhibition of nicotinic acetylcholine receptors by bicuculline

scientific article published in December 2001

Inhibition of nicotinic acetylcholine receptors by bicuculline is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0028-3908(01)00137-X
P698PubMed publication ID11684149

P50authorEleonora PalmaQ42816618
P2093author name stringMiledi R
Eusebi F
Demuro A
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Human neuronal threonine-for-leucine-248 alpha 7 mutant nicotinic acetylcholine receptors are highly Ca2+ permeableQ35119676
Ionic Blockage of Sodium Channels in NerveQ36388606
Modulation of nicotinic acetylcholine receptors by strychnineQ36459451
Neuronal nicotinic threonine-for-leucine 247 alpha7 mutant receptors show different gating kinetics when activated by acetylcholine or by the noncompetitive agonist 5-hydroxytryptamine.Q36578906
Strychnine activates neuronal alpha7 nicotinic receptors after mutations in the leucine ring and transmitter binding site domainsQ36676165
Threonine-for-leucine mutation within domain M2 of the neuronal alpha(7) nicotinic receptor converts 5-hydroxytryptamine from antagonist to agonist.Q37317700
Pharmacological characterization of different types of GABA and glutamate receptors in vertebrates and invertebrates☆☆☆Q38018942
The actions of picrotoxin, strychnine, bicuculline and other convulsants and antagonists on the responses to acetylcholine glutamic acid and gamma-aminobutyric acid on Helix neuronesQ39164397
A re-examination of curare action at the motor endplateQ39235257
GABA synaptic mechanisms: stereochemical and conformational requirementsQ39629796
Local anaesthetics transiently block currents through single acetylcholine-receptor channelsQ40676934
Bicuculline blocks nicotinic acetylcholine response in isolated intermediate lobe cells of the pigQ41932163
Glycine antagonists structurally related to 4,5,6,7-tetrahydroisoxazolo [5,4-c]pyridin-3-ol inhibit binding of [3H]strychnine to rat brain membranes.Q42038748
Effects of defolliculation on membrane current responses of Xenopus oocytesQ44580602
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Bicuculline and picrotoxin as antagonists of gamma-aminobutyrate and neuromuscular inhibition in the lobsterQ48554990
Bicuculline methiodide potentiates NMDA-dependent burst firing in rat dopamine neurons by blocking apamin-sensitive Ca2+-activated K+ currentsQ48646633
The specificity of strychnine as a glycine antagonist in the mammalian spinal cordQ48818882
Bicuculline and Central GABA ReceptorsQ48882915
A functional comparison of the antagonists bicuculline and picrotoxin at recombinant GABAA receptorsQ49023322
Bicuculline blocks the response to acetylcholine and nicotine but not to muscarine or GABA in isolated insect neuronal somata.Q52460665
Stereospecific interaction of bicuculline with specific [3H]strychnine binding to rat spinal cord synaptosomal membranesQ67288256
The action of bicuculline upon acetylcholine-induced excitations of central neuronesQ70055802
Cholinergic and catecholaminergic receptors in the Xenopus oocyte membraneQ70485790
Effects of 5-hydroxytryptamine on central neurones antagonized by bicuculline and picrotoxinQ70953086
Voltage dependence of mouse acetylcholine receptor gating: different charge movements in di-, mono- and unliganded receptorsQ71549837
A calcium-dependent transient outward current in Xenopus laevis oocytesQ72538085
P433issue7
P304page(s)854-861
P577publication date2001-12-01
P1433published inNeuropharmacologyQ15332439
P1476titleInhibition of nicotinic acetylcholine receptors by bicuculline
P478volume41

Reverse relations

cites work (P2860)
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