A novel structural class of potent inhibitors of NF-kappa B activation: structure-activity relationships and biological effects of 6-aminoquinazoline derivatives

scientific article published in September 2003

A novel structural class of potent inhibitors of NF-kappa B activation: structure-activity relationships and biological effects of 6-aminoquinazoline derivatives is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0968-0896(03)00438-3
P698PubMed publication ID12927847

P2093author name stringHideyuki Tomizawa
Hideya Hayashi
Yoshiaki Isobe
Masanori Tobe
Takahiro Nagasaki
Hirotada Takahashi
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Nuclear factor-kappa B is activated in alveolar macrophages from patients with acute respiratory distress syndrome.Q51023210
The mechanism of the inflammatory effect of carrageeninQ71109438
Novel inhibitors of cytokine-induced IkappaBalpha phosphorylation and endothelial cell adhesion molecule expression show anti-inflammatory effects in vivoQ73596145
Synthesis of NF-kappaB activation inhibitors derived from epoxyquinomicin CQ73895525
NF-kappa B activation in human knee-joint synovial tissue during the early stage of joint inflammationQ73921132
The NF-kappa B and I kappa B proteins: new discoveries and insightsQ24313579
Nuclear factor-kappaB: a pivotal transcription factor in chronic inflammatory diseasesQ29547555
NF-kappa B: ten years afterQ29618566
The effect of a T cell-specific NF-kappa B inhibitor on in vitro cytokine production and collagen-induced arthritisQ30886735
Local administration of transcription factor decoy oligonucleotides to nuclear factor-kappaB prevents carrageenin-induced inflammation in rat hind paw.Q38306587
Mechanistic aspects of NF-kappa B regulation: the emerging role of phosphorylation and proteolysisQ40410066
Inhibition of TNF-alpha-induced NF-kappaB activation and IL-8 release in A549 cells with the proteasome inhibitor MG-132.Q41017734
P433issue18
P407language of work or nameEnglishQ1860
P921main subjectNF-κBQ411114
P304page(s)3869-3878
P577publication date2003-09-01
P1433published inBioorganic & Medicinal ChemistryQ2904200
P1476titleA novel structural class of potent inhibitors of NF-kappa B activation: structure-activity relationships and biological effects of 6-aminoquinazoline derivatives
P478volume11

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