High-throughput cytochrome P450 inhibition screening via cassette probe-dosing strategy. IV. Validation of a direct injection on-line guard cartridge extraction/tandem mass spectrometry method for simultaneous CYP3A4, 2D6 and 2E1 inhibition assessme

scientific article published on 01 January 2000

High-throughput cytochrome P450 inhibition screening via cassette probe-dosing strategy. IV. Validation of a direct injection on-line guard cartridge extraction/tandem mass spectrometry method for simultaneous CYP3A4, 2D6 and 2E1 inhibition assessme is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1002/1097-0231(20001030)14:20<1943::AID-RCM116>3.0.CO;2-F
P698PubMed publication ID11013424

P2093author name stringP Teitelbaum
H Z Bu
K Knuth
L Magis
P2860cites workDetermination of a 'GW cocktail' of cytochrome P450 probe substrates and their metabolites in plasma and urine using automated solid phase extraction and fast gradient liquid chromatography tandem mass spectrometry.Q51432740
CYP2D6- and CYP3A-dependent metabolism of dextromethorphan in humansQ57314131
High-throughput caco-2 cell permeability screening by cassette dosing and sample pooling approaches using direct injection/on-line guard cartridge extraction/tandem mass spectrometryQ73549731
Validation of the five-drug "Pittsburgh cocktail" approach for assessment of selective regulation of drug-metabolizing enzymesQ73846452
Fully automated analysis of activities catalysed by the major human liver cytochrome P450 (CYP) enzymes: assessment of human CYP inhibition potentialQ74608267
Automated high throughput human CYP isoform activity assay using SPE-LC/MS method: application in CYP inhibition evaluationQ93930477
P433issue20
P304page(s)1943-1948
P577publication date2000-01-01
P1433published inRapid Communications in Mass SpectrometryQ3419582
P1476titleHigh-throughput cytochrome P450 inhibition screening via cassette probe-dosing strategy. IV. Validation of a direct injection on-line guard cartridge extraction/tandem mass spectrometry method for simultaneous CYP3A4, 2D6 and 2E1 inhibition assessment
P478volume14

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cites work (P2860)
Q73855267Current literature in mass spectrometry
Q44239831High-throughput inhibition screening of major human cytochrome P450 enzymes using an in vitro cocktail and liquid chromatography-tandem mass spectrometry
Q36716929Methods for predicting human drug metabolism
Q44194942Rapid and quantitative determination of metabolites from multiple cytochrome P450 probe substrates by gradient liquid chromatography-electrospray ionization-ion trap mass spectrometry

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