scholarly article | Q13442814 |
P50 | author | Claudiu T Supuran | Q28211545 |
Ahmed Elkamhawy | Q57012693 | ||
P2093 | author name string | Eun Joo Roh | |
So Ha Lee | |||
Wagdy M Eldehna | |||
Mohamed A Abdelgawad | |||
Silvia Bua | |||
Mohammad M Al-Sanea | |||
Sora Paik | |||
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Quinoline: a promising antitubercular target | Q38280178 | ||
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4-Aminoquinoline derivatives as novel Mycobacterium tuberculosis GyrB inhibitors: Structural optimization, synthesis and biological evaluation | Q38839891 | ||
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Antidepressant and antipsychotic activity of new quinoline- and isoquinoline-sulfonamide analogs of aripiprazole targeting serotonin 5-HT₁A/5-HT₂A/5-HT₇ and dopamine D₂/D₃ receptors | Q42713573 | ||
Carbonic anhydrase inhibitors | Q43042271 | ||
Carbonic anhydrase inhibitors: inhibition of mammalian isoforms I-XIV with a series of substituted phenols including paracetamol and salicylic acid | Q46519336 | ||
Synthesis of bulky-tailed sulfonamides incorporating pyrido[2,3-d][1,2,4]triazolo[4,3-a]pyrimidin-1(5H)-yl) moieties and evaluation of their carbonic anhydrases I, II, IV and IX inhibitory effects. | Q46697605 | ||
An Overview of the Bacterial Carbonic Anhydrases | Q47145746 | ||
Carbon- versus sulphur-based zinc binding groups for carbonic anhydrase inhibitors? | Q47692161 | ||
Discovery of curcumin inspired sulfonamide derivatives as a new class of carbonic anhydrase isoforms I, II, IX, and XII inhibitors | Q47719833 | ||
Quantitative assessment of specific carbonic anhydrase inhibitors effect on hypoxic cells using electrical impedance assays | Q47809412 | ||
Synthesis and biological evaluation of histamine Schiff bases as carbonic anhydrase I, II, IV, VII, and IX activators. | Q48000247 | ||
Synthesis and carbonic anhydrase I, II, VII, and IX inhibition studies with a series of benzo[d]thiazole-5- and 6-sulfonamides | Q48017394 | ||
3H-1,2-benzoxathiepine 2,2-dioxides: a new class of isoform-selective carbonic anhydrase inhibitors. | Q48030765 | ||
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Crystal structure of the human carbonic anhydrase II adduct with 1-(4-sulfamoylphenyl-ethyl)-2,4,6-triphenylpyridinium perchlorate, a membrane-impermeant, isoform selective inhibitor. | Q49332625 | ||
3D QSAR studies, pharmacophore modeling, and virtual screening of diarylpyrazole-benzenesulfonamide derivatives as a template to obtain new inhibitors, using human carbonic anhydrase II as a model protein. | Q51094113 | ||
Carbonic anhydrase activators. | Q51767411 | ||
2-Benzylpiperazine: A new scaffold for potent human carbonic anhydrase inhibitors. Synthesis, enzyme inhibition, enantioselectivity, computational and crystallographic studies and in vivo activity for a new class of intraocular pressure lowering age | Q52596189 | ||
Carbonic Anhydrases and Metabolism. | Q52645009 | ||
Antileishmanial activity of sulphonamide nanoemulsions targeting the β-carbonic anhydrase from Leishmania species. | Q55611103 | ||
Discovery of novel 1,3-diaryltriazene sulfonamides as carbonic anhydrase I, II, VII, and IX inhibitors | Q57279715 | ||
Quinoline and quinolone dimers and their biological activities: An overview | Q57814239 | ||
A Small-Molecule Drug Conjugate for the Treatment of Carbonic Anhydrase IX Expressing Tumors | Q57911941 | ||
Novel thiazolidinone-containing compounds, without the well-known sulphonamide zinc-binding group acting as human carbonic anhydrase IX inhibitors | Q58700155 | ||
Quinoline-Based p300 Histone Acetyltransferase Inhibitors with Pro-apoptotic Activity in Human Leukemia U937 Cells | Q58855679 | ||
Carbonic Anhydrase Inhibitors: Clash with Ala65 as a Means for Designing Inhibitors with Low Affinity for the Ubiquitous Isozyme II, Exemplified by the Crystal Structure of the Topiramate Sulfamide Analogue† | Q58863277 | ||
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A new approach to antiglaucoma drugs: carbonic anhydrase inhibitors with or without NO donating moieties. Mechanism of action and preliminary pharmacology | Q84679919 | ||
Synthesis, carbonic anhydrase I and II inhibition studies of the 1,3,5-trisubstituted-pyrazolines | Q88614584 | ||
Synthesis and pharmacological evaluation of pyrazolo[4,3-c]quinolinones as high affinity GABAA-R ligands and potential anxiolytics | Q89320179 | ||
Biomedical applications of prokaryotic carbonic anhydrases | Q89420700 | ||
Novel hydrazido benzenesulfonamides-isatin conjugates: Synthesis, carbonic anhydrase inhibitory activity and molecular modeling studies | Q90714675 | ||
Carbonic anhydrase inhibitors as antitumor/antimetastatic agents: a patent review (2008-2018) | Q90735662 | ||
Green recipes to quinoline: A review | Q90800498 | ||
Applications of carbonic anhydrases inhibitors in renal and central nervous system diseases | Q91269702 | ||
Carbonic anhydrase inhibitors and their potential in a range of therapeutic areas | Q91453043 | ||
Tumor-associated carbonic anhydrase isoform IX and XII inhibitory properties of certain isatin-bearing sulfonamides endowed with in vitro antitumor activity towards colon cancer | Q91467343 | ||
P275 | copyright license | Creative Commons Attribution 4.0 International | Q20007257 |
P6216 | copyright status | copyrighted | Q50423863 |
P433 | issue | 1 | |
P304 | page(s) | 1457-1464 | |
P577 | publication date | 2019-12-01 | |
P1433 | published in | Journal of Enzyme Inhibition and Medicinal Chemistry | Q15708877 |
P1476 | title | Synthesis and biological evaluation of novel 3-(quinolin-4-ylamino)benzenesulfonamidesAQ3 as carbonic anhydrase isoforms I and II inhibitors | |
P478 | volume | 34 |