Telacebec (Q203)-containing intermittent oral regimens sterilized mice infected with Mycobacterium ulcerans after only 16 doses

scientific article published on 31 August 2020

Telacebec (Q203)-containing intermittent oral regimens sterilized mice infected with Mycobacterium ulcerans after only 16 doses is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1371/JOURNAL.PNTD.0007857
P932PMC publication ID7494103
P698PubMed publication ID32866170

P50authorJerome RobertQ56858042
Aurélie ChauffourQ88580413
P2093author name stringVincent Jarlier
Kevin Pethe
Alexandra Aubry
Nicolas Veziris
P2860cites workDelayed versus standard assessment for excision surgery in patients with Buruli ulcer in Benin: a randomised controlled trial.Q54244183
Targeting the Mycobacterium ulcerans cytochrome bc:aa for the treatment of Buruli ulcerQ60020041
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Rifampicin and clarithromycin (extended release) versus rifampicin and streptomycin for limited Buruli ulcer lesions: a randomised, open-label, non-inferiority phase 3 trialQ90325404
Buruli ulcer treatment: Rate of surgical intervention differs highly between treatment centers in West AfricaQ90970892
Shortening Buruli Ulcer Treatment with Combination Therapy Targeting the Respiratory Chain and Exploiting Mycobacterium ulcerans Gene DecayQ91623033
Towards a new combination therapy for tuberculosis with next generation benzothiazinonesQ27681604
Benzothiazinones kill Mycobacterium tuberculosis by blocking arabinan synthesisQ28486345
In-vitro activity of avermectins against Mycobacterium ulceransQ28543887
Selamectin Is the Avermectin with the Best Potential for Buruli Ulcer TreatmentQ28547238
Efficacy of Rifampin Plus Clofazimine in a Murine Model of Mycobacterium ulcerans DiseaseQ28552524
Sterilizing Activity of Fully Oral Intermittent Regimens against Mycobacterium Ulcerans Infection in MiceQ28552736
Discovery of Q203, a potent clinical candidate for the treatment of tuberculosis.Q30352594
Bactericidal activity of rifampin-amikacin against Mycobacterium ulcerans in miceQ34144367
Single- and multiple-dose pharmacokinetics and absolute bioavailability of tedizolidQ34658779
In vitro and in vivo activities of rifampin, streptomycin, amikacin, moxifloxacin, R207910, linezolid, and PA-824 against Mycobacterium ulcerans.Q34680628
Potent twice-weekly rifapentine-containing regimens in murine tuberculosisQ35776635
Pharmacokinetics and pharmacodynamics of TMC207 and its N-desmethyl metabolite in a murine model of tuberculosisQ35806445
Comparative pharmacodynamics of the new oxazolidinone tedizolid phosphate and linezolid in a neutropenic murine Staphylococcus aureus pneumonia modelQ36364009
Anthelmintic avermectins kill Mycobacterium tuberculosis, including multidrug-resistant clinical strainsQ36558371
Bactericidal and sterilizing activities of several orally administered combined regimens against Mycobacterium ulcerans in miceQ36703065
Tedizolid (TR-701): a new oxazolidinone with enhanced potencyQ37983130
Tedizolid: The First Once-Daily Oxazolidinone Class AntibioticQ38536296
Intracellular activity of tedizolid phosphate and ACH-702 versus Mycobacterium tuberculosis infected macrophagesQ38749324
THE EXPERIMENTAL DISEASE THAT FOLLOWS THE INJECTION OF HUMAN LEPROSY BACILLI INTO FOOT-PADS OF MICE.Q41861671
Brain penetration of ivermectin and selamectin in mdr1a,b P-glycoprotein- and bcrp- deficient knockout miceQ46152205
DprE1, a new taxonomic marker in mycobacteriaQ48037784
P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P433issue8
P921main subjectMycobacterium ulceransQ141154
P304page(s)e0007857
P577publication date2020-08-31
P1433published inPLoS Neglected Tropical DiseasesQ3359737
P1476titleTelacebec (Q203)-containing intermittent oral regimens sterilized mice infected with Mycobacterium ulcerans after only 16 doses
P478volume14