Subtype selective binding properties of substituted linear melanocyte stimulating hormone analogues

scientific article

Subtype selective binding properties of substituted linear melanocyte stimulating hormone analogues is …
instance of (P31):
scholarly articleQ13442814

External links are
P356DOI10.1016/S0143-4179(02)00133-6
P698PubMed publication ID12507437

P50authorHelgi B. SchiöthQ30112644
P2093author name stringJarl E S Wikberg
Ilze Mutule
Hajime Watanobe
Ruta Muceniece
Felikss Mutulis
Aster Tesfaye
Richard Rudzish
P2860cites workMolecular cloning of a novel human melanocortin receptorQ28263897
Discovery of novel melanocortin4receptor selective MSH analoguesQ29026417
Synthesis of 153N-6 analogues and structure-function analysis at murine melanocortin-1 (MC1) receptorsQ30634375
New aspects on the melanocortins and their receptorsQ30939118
Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH(2) at the mouse melanocortin receptors. 1. Modifications at the His positionQ31076926
Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH(2) at the mouse melanocortin receptors: part 2 modifications at the Phe positionQ31089001
Selective properties of C- and N-terminals and core residues of the melanocyte-stimulating hormone on binding to the human melanocortin receptor subtypesQ32052313
Melanocortins and the brain: from effects via receptors to drug targetsQ34060958
The physiological role of melanocortin receptorsQ34254198
Discovery of Prototype Peptidomimetic Agonists at the Human Melanocortin Receptors MC1R and MC4RQ36870130
Selectivity of cyclic [D-Nal7] and [D-Phe7] substituted MSH analogues for the melanocortin receptor subtypesQ36889306
Novel cyclic templates of alpha-MSH give highly selective and potent antagonists/agonists for human melanocortin-3/4 receptorsQ40728850
D-Amino acid scan of gamma-melanocyte-stimulating hormone: importance of Trp(8) on human MC3 receptor selectivityQ40833260
The melanocortin (MC3) receptor from rat hypothalamus: photoaffinity labelling and binding of alanine-substituted alpha-MSH analoguesQ41448305
Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA.Q43581712
Synthesis and biological evaluation on hMC3, hMC4 and hMC5 receptors of gamma-MSH analogs substituted with L-alanineQ43967457
Modeling of the three-dimensional structure of the human melanocortin 1 receptor, using an automated method and docking of a rigid cyclic melanocyte-stimulating hormone core peptideQ47926577
Conformation of the core sequence in melanocortin peptides directs selectivity for the melanocortin MC3 and MC4 receptorsQ48192978
Asp10 in Lys-gamma2-MSH determines selective activation of the melanocortin MC3 receptorQ48401331
Characterization of melanocortin NDP-MSH agonist peptide fragments at the mouse central and peripheral melanocortin receptorsQ48845749
Design in topographical space of peptide and peptidomimetic ligands that affect behavior. A chemist's glimpse at the mind--body problem.Q52279728
Molecular Basis for the Interaction of [Nle4,d-Phe7]Melanocyte Stimulating Hormone with the Human Melanocortin-1 Receptor (Melanocyte α-MSH Receptor)Q57981267
Characterisation of the melanocortin 4 receptor by radioligand bindingQ71712692
Characterisation of melanocortin receptor subtypes by radioligand binding analysisQ72296957
Synthesis and biological evaluation of alpha-MSH analogues substituted with alanineQ72542949
Selectivity of [Phe-I7], [Ala6], and [D-Ala4,Gln5,Tyr6] substituted ACTH(4-10) analogues for the melanocortin receptorsQ73489059
Discovery and development of novel melanogenic drugs. Melanotan-I and -IIQ77370427
P433issue6
P304page(s)427-434
P577publication date2002-12-01
P1433published inNeuropeptidesQ15751202
P1476titleSubtype selective binding properties of substituted linear melanocyte stimulating hormone analogues
P478volume36

Reverse relations

Q41165076Comparative Functional Alanine Positional Scanning of the α-Melanocyte Stimulating Hormone and NDP-Melanocyte Stimulating Hormone Demonstrates Differential Structure-Activity Relationships at the Mouse Melanocortin Receptors.cites workP2860

Search more.