Selectivity of cyclic [D-Nal7] and [D-Phe7] substituted MSH analogues for the melanocortin receptor subtypes

scientific article published on January 1997

Selectivity of cyclic [D-Nal7] and [D-Phe7] substituted MSH analogues for the melanocortin receptor subtypes is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0196-9781(97)00079-X
P698PubMed publication ID9357059

P50authorHelgi B. SchiöthQ30112644
P2093author name stringHruby VJ
Sharma SD
Lindeberg G
Wikberg JE
Prusis P
Mutulis F
Müceniece R
P2860cites workThe cloning of a family of genes that encode the melanocortin receptorsQ24337156
Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionQ27860958
Molecular cloning of a novel human melanocortin receptorQ28263897
Evaluation of melanotan-II, a superpotent cyclic melanotropic peptide in a pilot phase-I clinical studyQ28279545
4-Norleucine, 7-D-phenylalanine-alpha-melanocyte-stimulating hormone: a highly potent alpha-melanotropin with ultralong biological activityQ28367158
half-Cys4,half-Cys10-alpha-Melanocyte-stimulating hormone: a cyclic alpha-melanotropin exhibiting superagonist biological activityQ36286550
Regulation of the synthesis of steroidogenic enzymes in adrenal cortical cells by ACTH.Q39216606
The opiomelanotropinergic neuronal and endocrine systemsQ40131246
Expression of functional melanocortin 1 receptors in insect cellsQ41204619
Major pharmacological distinction of the ACTH receptor from other melanocortin receptorsQ41250598
Cyclic lactam alpha-melanotropin analogues of Ac-Nle4-cyclo[Asp5, D-Phe7,Lys10] alpha-melanocyte-stimulating hormone-(4-10)-NH2 with bulky aromatic amino acids at position 7 show high antagonist potency and selectivity at specific melanocortin recepQ41301816
The melanocortin (MC3) receptor from rat hypothalamus: photoaffinity labelling and binding of alanine-substituted alpha-MSH analoguesQ41448305
Molecular cloning and expression of the human melanocyte stimulating hormone receptor cDNA.Q43581712
A three dimensional model for the interaction of MSH with the melanocortin-1 receptorQ49270179
Potent and prolonged acting cyclic lactam analogues of alpha-melanotropin: design based on molecular dynamicsQ69360120
Cyclic melanotropins. 5. Importance of the C-terminal tripeptide (Lys-Pro-Val)Q70223708
Structure-activity studies of highly potent cyclic [Cys4,Cys10]Melanotropin analoguesQ70983217
Characterisation of the melanocortin 4 receptor by radioligand bindingQ71712692
Characterisation of melanocortin receptor subtypes by radioligand binding analysisQ72296957
Synthesis and biological evaluation of alpha-MSH analogues substituted with alanineQ72542949
P433issue7
P304page(s)1009-1013
P577publication date1997-01-01
P1433published inPeptidesQ7166533
P1476titleSelectivity of cyclic [D-Nal7] and [D-Phe7] substituted MSH analogues for the melanocortin receptor subtypes
P478volume18

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