Aminoglycosides: activity and resistance

scientific article

Aminoglycosides: activity and resistance is …
instance of (P31):
review articleQ7318358
scholarly articleQ13442814

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P356DOI10.1128/AAC.43.4.727
P932PMC publication ID89199
P698PubMed publication ID10103173

P2093author name stringP M Tulkens
M P Mingeot-Leclercq
Y Glupczynski
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Antibacterial activity and ototoxicity in guinea pigs, and nephrotoxicity in rats of arbekacin.Q53885852
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Synthesis of dibekacin analogs containing 3-oxa- and 3-aza-2,3,4-trideoxy-D-glycero-hexopyranose.Q53980687
A synthetic study of methyl 3-deoxy-3-fluoro-alpha-D-glucopyranosides from methyl 2,3-anhydro-alpha-D-allopyranosides, and synthesis of 3'-deoxy-3'-fluorokanamycin A and 3'-chloro-3'-deoxykanamycin AQ54067249
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Active-site labeling of an aminoglycoside antibiotic phosphotransferase (APH(3')-IIIa).Q54190990
Susceptibility of methicillin-resistant Staphylococcus aureus clinical isolates to various antimicrobial agents. IV. Aminoglycoside-modifying enzyme AAC(6')/APH(2") is responsible for arbekacin-resistance enhanced by bleomycin.Q54196937
Structures of enzymatically modified products of arbekacin by methicillin-resistant. Staphylococcus aureus.Q54247959
New derivatives of kanamycin B obtained by combined modifications in positions 1 and 6". Synthesis, microbiological properties, and in vitro and computer-aided toxicological evaluation.Q54298674
Synthesis of 3'-deoxy-3'-fluorokanamycin A and 3',4'-dideoxy-3'-fluorokanamycin A.Q54299872
Resistance to aminoglycoside antibiotics in gram-negative bacilli and staphylococci isolated from blood. Report from a European collaborative study. The ESGAR Study Group (European Study Group on Antibiotic Resistance).Q54320617
Substrate specificities and structure-activity relationships for the nucleotidylation of antibiotics catalyzed by aminoglycoside nucleotidyltransferase 2''-I.Q54383442
Synthesis of 3'-deoxy-3'-fluorokanamycins A and B active against resistant bacteria.Q54444543
Expression of prokaryotic genes for hygromycin B and G418 resistance as dominant-selection markers in mouse L cellsQ54468305
Structure-activity relationships of hygromycin A and its analogs: protein synthesis inhibition activity in a cell free system.Q54564545
3',4'-dideoxy-kanamycin B active against kanamycin-resistant Escherichia coli and Pseudomonas aeruginosaQ54668246
Altered denA and anr gene expression in aminoglycoside adaptive resistance in Pseudomonas aeruginosaQ57238285
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Synthesis of 5-deoxy-5-fluoro and 5-deoxy-5,5-difluoro derivatives of kanamycin B and its analogs. Study on structure-toxicity relationshipsQ67573571
A synthesis of 3',4'-dideoxykanamycin BQ67809653
In vitro susceptibility to aminoglycoside antibiotics in blood and urine isolates consecutively collected in twenty-nine European laboratories. European Study Group on Antibiotic ResistanceQ68194936
Aminoglycoside antibiotic treatment of human fibroblasts: intracellular accumulation, molecular changes and the loss of ribosomal accuracyQ68988579
Aminoglycoside antibiotics. II. Configurational and positional isomers of BB-K8Q69661389
Letter: Syntheses of 1-n-(S)-4-amino-2-hydroxybutyryl)-kanamycin B and -3', 4'-dideoxykanamycin B active against kanamycin-resistant bacteriaQ69662851
Determination of the rate-limiting segment of aminoglycoside nucleotidyltransferase 2''-I by pH and viscosity-dependent kineticsQ69835168
Interaction of gentamicin and spermine with bilayer membranes containing negatively charged phospholipidsQ70069613
Chemical modification of amikacin at C-4'' with inversion of configurationQ70111368
Biphasic, concentration-dependent and rate-limited, concentration-independent bacterial killing by an aminoglycoside antibioticQ70502539
Synthesis of low-toxicity, 5-deoxy-5-fluoro and 5-deoxy-5,5-difluoro derivatives of arbekacin and its analogs, and study of structure-toxicity relationshipsQ70622908
New 2''-amino derivatives of arbekacin, potent aminoglycoside antibiotics against methicillin-resistant Staphylococcus aureusQ70671045
The most frequently occurring aminoglycoside resistance mechanisms--combined results of surveys in eight regions of the world. The Aminoglycoside Resistance Study GroupsQ71059885
Studies on a new aminoglycoside antibiotic, dactimicin. II. Isolation, structure and chemical degradationQ71066927
A prospective, randomized study of amikacin and gentamicin in serious infections with focus on efficacy, toxicity and duration of serum levels above the MICQ71104190
Enzymatic 2'-N-acetylation of arbekacin and antibiotic activity of its productQ71195666
Selective elimination of fibroblasts from cultures of normal human melanocytesQ71355336
Synthesis and antimicrobial and toxicological studies of amino acid and peptide derivatives of kanamycin A and netilmicinQ71514431
Specificity of aminoglycoside binding to RNA constructs derived from the 16S rRNA decoding region and the HIV-RRE activator regionQ73040655
P433issue4
P407language of work or nameEnglishQ1860
P304page(s)727-737
P577publication date1999-04-01
P1433published inAntimicrobial Agents and ChemotherapyQ578004
P1476titleAminoglycosides: activity and resistance
P478volume43

Reverse relations

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Q50484768[Aminoglycosides].
Q42184041armA and aminoglycoside resistance in Escherichia coli
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