scholarly article | Q13442814 |
P2093 | author name string | Jing Zhang | |
Bin Wang | |||
Dominic Ryan | |||
Anu Daniel | |||
Blaise Lippa | |||
Brian Chamberlain | |||
Chester A Metcalf | |||
Douglas Bevan | |||
Felix Epie | |||
Jan Antoinette C Romero | |||
Jared Silverman | |||
Joseph Shotwell | |||
Katherine M Poutsiaka | |||
Kien Nguyen | |||
Nicole Carter | |||
Qingyi Yang | |||
Roland E Dolle | |||
Terence Moy | |||
Vipul Kumar | |||
Jason Cross | |||
Anu Arya | |||
Yuchuan Wu | |||
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Novel inhibitors of DNA gyrase: 3D structure based biased needle screening, hit validation by biophysical methods, and 3D guided optimization. A promising alternative to random screening | Q31406783 | ||
Exploiting bacterial DNA gyrase as a drug target: current state and perspectives. | Q34214929 | ||
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Prospects for developing new antibacterials targeting bacterial type IIA topoisomerases. | Q38162903 | ||
The nature of inhibition of DNA gyrase by the coumarins and the cyclothialidines revealed by X-ray crystallography | Q41064279 | ||
5-(2-Pyrimidinyl)-imidazo[1,2-a]pyridines are antibacterial agents targeting the ATPase domains of DNA gyrase and topoisomerase IV. | Q43291231 | ||
Novel dual-targeting benzimidazole urea inhibitors of DNA gyrase and topoisomerase IV possessing potent antibacterial activity: intelligent design and evolution through the judicious use of structure-guided design and structure-activity relationship | Q44006954 | ||
Structure-activity relationship (SAR): effort towards blocking N-glucuronidation of indazoles (PF-03376056) by human UGT1A enzymes | Q46056539 | ||
A new DNA gyrase inhibitor subclass of the cyclothialidine family based on a bicyclic dilactam-lactone scaffold. Synthesis and antibacterial properties | Q83570903 | ||
P433 | issue | 10 | |
P304 | page(s) | 1080-1085 | |
P577 | publication date | 2015-09-08 | |
P1433 | published in | ACS Medicinal Chemistry Letters | Q2819061 |
P1476 | title | Discovery of Indazole Derivatives as a Novel Class of Bacterial Gyrase B Inhibitors | |
P478 | volume | 6 |
Q48266288 | Design, Synthesis, and Evaluation of Novel Tyrosine-Based DNA Gyrase B Inhibitors. |
Q35994500 | Discovery of Pyrazolopyridones as a Novel Class of Gyrase B Inhibitors Using Structure Guided Design |
Q57265865 | New N-phenylpyrrolamide DNA gyrase B inhibitors: Optimization of efficacy and antibacterial activity |
Q91666978 | Synthesis and biological evaluation against Leishmania donovani of novel hybrid molecules containing indazole-based 2-pyrone scaffolds |
Q46478240 | Targeting DNA Replication and Repair for the Development of Novel Therapeutics against Tuberculosis |
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