MCR synthesis of praziquantel derivatives

scientific article published on 30 January 2012

MCR synthesis of praziquantel derivatives is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1111/J.1747-0285.2011.01288.X
P932PMC publication ID3712825
P698PubMed publication ID22151001

P50authorAlex DomlingQ73024340
P2093author name stringHaixia Liu
Sanaa Botros
Eberhardt Herdtweck
Samia William
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Synthesis and properties of Praziquantel, a novel broad spectrum anthelmintic with excellent activity against Schistosomes and CestodesQ56656937
Cyclizations ofN-Acyliminium IonsQ56831862
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Praziquantel: mechanisms of action, resistance and new derivatives for schistosomiasisQ37315241
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Synthesis, biological evaluation, and molecular docking of Ugi products containing a zinc-chelating moiety as novel inhibitors of histone deacetylases.Q39864415
Efficient multicomponent reaction synthesis of the schistosomiasis drug praziquantel.Q42906063
Efficient and diverse synthesis of indole derivatives.Q43296555
Amino acid derived heterocycles: lewis acid catalyzed and radical cyclizations from peptide acetalsQ44021182
Effect of praziquantel on the immature stages of Schistosoma haematobium.Q46588110
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An Improved Perfusion Technique for Recovering Adult Schistosomes from Laboratory AnimalsQ53755844
P433issue4
P921main subjectpraziquantelQ424145
P304page(s)470-477
P577publication date2012-01-30
P1433published inChemical Biology and Drug DesignQ15749458
P1476titleMCR synthesis of praziquantel derivatives
P478volume79

Reverse relations

cites work (P2860)
Q28539960'Death and axes': unexpected Ca²⁺ entry phenologs predict new anti-schistosomal agents
Q46836910Artificial Macrocycles by Ugi Reaction and Passerini Ring Closure.
Q38067995Ca²⁺ channels and praziquantel: a view from the free world
Q89920010Current and Novel Therapies Against Helminthic Infections: The Potential of Antioxidants Combined with Drugs
Q64082229Diverse Isoquinoline Scaffolds by Ugi/Pomeranz-Fritsch and Ugi/Schlittler-Müller Reactions
Q52699502Drug Repurposing for Schistosomiasis: Combinations of Drugs or Biomolecules.
Q28547995Ergot Alkaloids (Re)generate New Leads as Antiparasitics
Q64077252MCR Scaffolds Get Hotter with F-Labeling
Q36522303MCR synthesis of a tetracyclic tetrazole scaffold.
Q34060368Modern Multicomponent Reactions for better Drug Syntheses**
Q27008897Novel therapeutic and prevention approaches for schistosomiasis: review
Q39160696Praziquantel derivatives with antischistosomal activity: aromatic ring modification
Q46081944Synthesis and SAR studies of praziquantel derivatives with activity against Schistosoma japonicum.
Q61802827Tetrazoles via Multicomponent Reactions
Q92815392The Pictet-Spengler Reaction Updates Its Habits
Q42550963Tricycles by a new Ugi variation and Pictet-Spengler reaction in one pot.
Q42612607Various cyclization scaffolds by a truly Ugi 4-CR.
Q45340054[(η(6)-Praziquantel)Cr(CO)3] derivatives with remarkable in vitro anti-schistosomal activity

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