review article | Q7318358 |
scholarly article | Q13442814 |
P2093 | author name string | Iwan J P de Esch | |
Rob Leurs | |||
Paul L Chazot | |||
Fiona C Shenton | |||
Herman D Lim | |||
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Characterization of the histamine H4 receptor binding site. Part 1. Synthesis and pharmacological evaluation of dibenzodiazepine derivatives | Q40253729 | ||
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Identification of rat H3 receptor isoforms with different brain expression and signaling properties. | Q43513207 | ||
The role of transmembrane helix 5 in agonist binding to the human H3 receptor | Q43964575 | ||
Immunohistochemical localization of histamine receptor subtypes in human inferior turbinates | Q44993372 | ||
Localization of histamine H4 receptors in the central nervous system of human and rat. | Q46153368 | ||
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Comparative study of histamine H4 receptor expression in human dermal fibroblasts | Q46338219 | ||
Rotationally constrained 2,4-diamino-5,6-disubstituted pyrimidines: a new class of histamine H4 receptor antagonists with improved druglikeness and in vivo efficacy in pain and inflammation models | Q46347020 | ||
Histamine H4 receptors modulate dendritic cell migration through skin--immunomodulatory role of histamine | Q46377867 | ||
Histamine H4 receptor stimulation suppresses IL-12p70 production and mediates chemotaxis in human monocyte-derived dendritic cells | Q46448103 | ||
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Histamine H3 and H4 receptors are expressed on distinct endocrine cell types in the rat fundic mucosa | Q46697957 | ||
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Auto-inhibition of brain histamine release mediated by a novel class (H3) of histamine receptor | Q34249836 | ||
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P433 | issue | 1 | |
P407 | language of work or name | English | Q1860 |
P921 | main subject | pharmacology | Q128406 |
P304 | page(s) | 14-23 | |
P577 | publication date | 2009-05-01 | |
P1433 | published in | British Journal of Pharmacology | Q919631 |
P1476 | title | Molecular and biochemical pharmacology of the histamine H4 receptor | |
P478 | volume | 157 |
Q58694870 | A Selective Histamine H Receptor Antagonist, JNJ7777120, Is Protective in a Rat Model of Transient Cerebral Ischemia |
Q48491449 | A search for functional histamine H4 receptors in the human, guinea pig and mouse brain |
Q43110514 | Advances in histamine pharmacology reveal new drug targets |
Q37553620 | Aryl-1,3,5-triazine ligands of histamine H4 receptor attenuate inflammatory and nociceptive response to carrageen, zymosan and lipopolysaccharide |
Q37551908 | Biased G Protein-Coupled Receptor Signaling: New Player in Modulating Physiology and Pathology |
Q39445688 | Commercially available antibodies against human and murine histamine H₄-receptor lack specificity |
Q42020167 | Comparison of the pharmacological properties of human and rat histamine H3-receptors |
Q38152336 | Current and emerging options for the drug treatment of narcolepsy |
Q39204577 | Detailed analysis of biased histamine H₄ receptor signalling by JNJ 7777120 analogues |
Q39323929 | Development of a profiling strategy for metabolic mixtures by combining chromatography and mass spectrometry with cell-based GPCR signaling |
Q47845214 | Effects of histamine H4 receptor ligands in a mouse model of gastric ulceration. |
Q38160491 | Eosinophils and mast cells as therapeutic targets in pediatric functional dyspepsia |
Q39584467 | Expression and functional properties of canine, rat, and murine histamine H₄ receptors in Sf9 insect cells. |
Q42182992 | Facilitation of short-term memory by histaminergic neurons in the nucleus accumbens is independent of cholinergic and glutamatergic transmission |
Q42951309 | GPCR theme editorial |
Q37598261 | Histamine H3 and H4 receptors as novel drug targets. |
Q38023551 | Histamine H3 receptor antagonists in relation to epilepsy and neurodegeneration: a systemic consideration of recent progress and perspectives. |
Q39166397 | Histamine H4 receptor agonist-induced relief from painful peripheral neuropathy is mediated by inhibition of spinal neuroinflammation and oxidative stress |
Q33752485 | Histamine H4 receptor antagonism inhibits allergen-specific T-cell responses mediated by human dendritic cells |
Q34025192 | Histamine H4 receptor as a new therapeutic target for choroidal neovascularization in age-related macular degeneration |
Q38264340 | Histamine H₄ receptors in the gastrointestinal tract. |
Q26799561 | Histamine and Skin Barrier: Are Histamine Antagonists Useful for the Prevention or Treatment of Atopic Dermatitis? |
Q26798112 | Histamine and the striatum |
Q38024865 | Histamine in brain development |
Q39639684 | Histamine modulates γδ-T lymphocyte migration and cytotoxicity, via Gi and Gs protein-coupled signalling pathways. |
Q37954375 | Histamine pharmacology and new CNS drug targets. |
Q34356076 | Histamine receptors and cancer pharmacology |
Q33688711 | Histamine therapeutic efficacy in metastatic melanoma: Role of histamine H4 receptor agonists and opportunity for combination with radiation. |
Q33574684 | Histamine: a new immunomodulatory player in the neuron-glia crosstalk |
Q37995651 | Histamine: an undercover agent in multiple rare diseases? |
Q64059638 | Human β-Defensin 2 Expression in Oral Epithelium: Potential Therapeutic Targets in Oral Lichen Planus |
Q90399887 | Influence of the Novel Histamine H3 Receptor Antagonist/Inverse Agonist M39 on Gastroprotection and PGE2 Production Induced by (R)-Alpha-Methylhistamine in C57BL/6 Mice |
Q41684431 | Lack of Histamine H4-Receptor Expression Aggravates TNBS-Induced Acute Colitis Symptoms in Mice. |
Q28536518 | Luciferase reporter gene assay on human, murine and rat histamine H4 receptor orthologs: correlations and discrepancies between distal and proximal readouts |
Q91871611 | Mast Cells May Differentially Regulate Growth of Lymphoid Neoplasms by Opposite Modulation of Histamine Receptors |
Q42554178 | Molecular determinants for the high constitutive activity of the human histamine H4 receptor: functional studies on orthologues and mutants |
Q92970095 | Pathophysiological Role of Histamine H4 Receptor in Cancer: Therapeutic Implications |
Q50875481 | Pharmacological targeting of histamine H4 receptor in periodontal disease. |
Q35161152 | Physiological implications of biased signaling at histamine H2 receptors |
Q34902203 | Protection of radiation-induced damage to the hematopoietic system, small intestine and salivary glands in rats by JNJ7777120 compound, a histamine H4 ligand. |
Q39498635 | Role of the second and third extracellular loops of the histamine H(4) receptor in receptor activation |
Q37944920 | Several down, a few to go: histamine H3 receptor ligands making the final push towards the market? |
Q64061747 | Structure-Activity Relationship of Hetarylpropylguanidines Aiming at the Development of Selective Histamine Receptor Ligands |
Q43097783 | TRPV1 and PLC Participate in Histamine H4 Receptor-Induced Itch |
Q58785720 | The Role of Histamine and Histamine Receptors in Mast Cell-Mediated Allergy and Inflammation: The Hunt for New Therapeutic Targets |
Q54383765 | The expression of histamine H4 receptor mRNA in the skin and other tissues of normal dogs. |
Q37151169 | Therapeutic potential of histamine H₄ receptor agonists in triple-negative human breast cancer experimental model. |