scholarly article | Q13442814 |
P356 | DOI | 10.1002/ANIE.201102965 |
P698 | PubMed publication ID | 21905185 |
P50 | author | Herbert Waldmann | Q1609256 |
Robin S. Bon | Q39476848 | ||
Frank J Dekker | Q39476878 | ||
P2093 | author name string | Stefan Wetzel | |
Steffen Renner | |||
Christian Hedberg | |||
Claas Gerding-Reimers | |||
Nachiket Vartak | |||
Philippe I H Bastiaens | |||
Marion Rusch | |||
P2860 | cites work | Small-molecule inhibition of APT1 affects Ras localization and signaling | Q24307840 |
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An acylation cycle regulates localization and activity of palmitoylated Ras isoforms | Q28306968 | ||
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Lipidated ras and rab peptides and proteins--synthesis, structure, and function | Q36619526 | ||
A functional screen implicates microRNA-138-dependent regulation of the depalmitoylation enzyme APT1 in dendritic spine morphogenesis | Q36678825 | ||
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Ras-MAPK pathway as a therapeutic target in cancer--emphasis on bladder cancer. | Q37516197 | ||
N-terminally myristoylated Ras proteins require palmitoylation or a polybasic domain for plasma membrane localization | Q38306703 | ||
H-ras but not K-ras traffics to the plasma membrane through the exocytic pathway | Q39451813 | ||
Thioesterase activity and subcellular localization of acylprotein thioesterase 1/lysophospholipase 1. | Q39852136 | ||
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Enzymatic depalmitoylation of viral glycoproteins with acyl-protein thioesterase 1 in vitro | Q40781982 | ||
Cloning, expression, and catalytic mechanism of murine lysophospholipase I. | Q41110642 | ||
Purification and properties of lysophospholipase isoenzymes from pig gastric mucosa | Q42160571 | ||
Regiospecificity and catalytic triad of lysophospholipase I. | Q43501837 | ||
Boron-mediated aldol reaction of carboxylic esters: complementary anti- and syn-selective asymmetric aldol reactions | Q44069924 | ||
Lysophospholipase I identified as a ghrelin deacylation enzyme in rat stomach | Q45157348 | ||
Beta-lactone probes identify a papain-like peptide ligase in Arabidopsis thaliana. | Q46460108 | ||
Lipidierte Ras- und Rab-Peptide und -Proteine: Synthese, Struktur und Funktion | Q57531482 | ||
P433 | issue | 42 | |
P407 | language of work or name | English | Q1860 |
P921 | main subject | protein design | Q410814 |
P304 | page(s) | 9832-9837 | |
P577 | publication date | 2011-09-09 | |
P1433 | published in | Angewandte Chemie International Edition | Q62023953 |
P1476 | title | Development of highly potent inhibitors of the Ras-targeting human acyl protein thioesterases based on substrate similarity design | |
P478 | volume | 50 |
Q52350987 | Acanthamoeba and Dictyostelium as Cellular Models for Legionella Infection. |
Q90434318 | Activity-Based Sensing of S-Depalmitoylases: Chemical Technologies and Biological Discovery |
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Q47445934 | Biodegradable zwitterionic sulfobetaine polymer and its conjugate with paclitaxel for sustained drug delivery. |
Q34317561 | Boron-based inhibitors of acyl protein thioesterases 1 and 2. |
Q28534102 | Cellular FRET-Biosensors to Detect Membrane Targeting Inhibitors of N-Myristoylated Proteins |
Q42028708 | Characterization of a serine hydrolase targeted by acyl-protein thioesterase inhibitors in Toxoplasma gondii |
Q34266996 | Chemical-biological exploration of the limits of the Ras de- and repalmitoylating machinery |
Q34785627 | Combining cross-metathesis and activity-based protein profiling: new β-lactone motifs for targeting serine hydrolases |
Q38534932 | Current status of the development of Ras inhibitors |
Q45228186 | Development of an activity-based probe and in silico design reveal highly selective inhibitors for diacylglycerol lipase-α in brain |
Q28533449 | Exploring anti-bacterial compounds against intracellular Legionella |
Q36957153 | Fat chance! Getting a grip on a slippery modification |
Q30844739 | Individual S-acylated cysteines differentially contribute to H-Ras endomembrane trafficking and acylation/deacylation cycles |
Q38802497 | Molecular Mechanism for Isoform-Selective Inhibition of Acyl Protein Thioesterases 1 and 2 (APT1 and APT2). |
Q42578090 | Multiexcitation Fluorogenic Labeling of Surface, Intracellular, and Total Protein Pools in Living Cells |
Q100156054 | Palmostatin B binds RAS depalmitoylases |
Q38568187 | Pharmacological Inhibition of Protein Lipidation |
Q47223139 | Posttranslational Modifications of RAS Proteins. |
Q36673837 | Profiling and inhibiting reversible palmitoylation |
Q47239374 | Protein Lipidation: Occurrence, Mechanisms, Biological Functions, and Enabling Technologies |
Q47295054 | Protein depalmitoylases. |
Q35188280 | Small-molecule modulation of Ras signaling |
Q41107898 | Spatial cycles mediated by UNC119 solubilisation maintain Src family kinases plasma membrane localisation |
Q39392568 | Synthesis and biological investigation of the β-thiolactone and β-lactam analogs of tetrahydrolipstatin |
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Q38423044 | Targeting RAS Membrane Association: Back to the Future for Anti-RAS Drug Discovery? |
Q36352506 | Targeting oncogenic Ras signaling in hematologic malignancies |
Q38223437 | Targeting protein palmitoylation: selective inhibitors and implications in disease |
Q44175173 | The mechanism of caseinolytic protease (ClpP) inhibition |
Q34003766 | Ultrafluorogenic coumarin-tetrazine probes for real-time biological imaging. |
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