Cloning, pharmacological characterisation and tissue distribution of a novel 5-HT4 receptor splice variant, 5-HT4(i).

scientific article published on 30 April 2004

Cloning, pharmacological characterisation and tissue distribution of a novel 5-HT4 receptor splice variant, 5-HT4(i). is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1007/S00210-004-0919-4
P698PubMed publication ID15118808

P2093author name stringAlberto J Kaumann
Finn Olav Levy
Trond Brattelid
Marit E Hystad
Kurt A Krobert
Trond Bach
Ane M Kvingedal
Kjetil W Andressen
P2860cites workCloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminusQ24319843
Cloning and expression of human 5-HT4S receptors. Effect of receptor density on their coupling to adenylyl cyclaseQ24322673
Isolation of the serotoninergic 5-HT4(e) receptor from human heart and comparative analysis of its pharmacological profile in C6-glial and CHO cell linesQ24675224
Relationship between the inhibition constant (K1) and the concentration of inhibitor which causes 50 per cent inhibition (I50) of an enzymatic reactionQ27860958
Molecular and functional characterization of a 5-HT4 receptor cloned from human atriumQ28116102
Absolute quantification of mRNA using real-time reverse transcription polymerase chain reaction assaysQ28140044
The 5-HT4 receptor: molecular cloning and pharmacological characterization of two splice variantsQ28368220
Structure of the human serotonin 5-HT4 receptor gene and cloning of a novel 5-HT4 splice variantQ28369138
Novel brain-specific 5-HT4 receptor splice variants show marked constitutive activity: role of the C-terminal intracellular domainQ28574308
Cloning and expression of a human serotonin 5-HT4 receptor cDNAQ28611165
Real-time RT-PCR for the detection of beta-adrenoceptor messenger RNAs in small human endomyocardial biopsies.Q30773692
5HT4(a) and 5-HT4(b) receptors have nearly identical pharmacology and are both expressed in human atrium and ventricleQ32059490
Quantitative mRNA analysis of five C-terminal splice variants of the human 5-HT4 receptor in the central nervous system by TaqMan real time RT-PCR.Q33951364
Structural and functional features of eukaryotic mRNA untranslated regionsQ33955093
Cloning and characterization of a novel human 5-HT4 receptor variant that lacks the alternatively spliced carboxy terminal exon. RT-PCR distribution in human brain and periphery of multiple 5-HT4 receptor variantsQ34105746
Do human atrial 5-HT4 receptors mediate arrhythmias?Q40610626
In situ assay of hormone-stimulated adenylyl cyclase in 96-well microtitration plates: an aide to rapid identification of transformed cell clonesQ41582953
Hormone-stimulated desensitization of hormone-dependent adenylyl cyclase. Dual action of luteninizing hormone on pig graafian follicle membranesQ42443756
An improved in vitro bioassay for the study of 5-HT(4) receptors in the human isolated large intestinal circular muscleQ43263780
Unaltered agonist potency upon inducible 5-HT7(a) but not 5-HT4(b) receptor expression indicates agonist-independent association of 5-HT7(a) receptor and Gs.Q44548147
A highly sensitive adenylate cyclase assayQ47871494
Comparison of the densities of 5-HT4 receptors, beta 1- and beta 2-adrenoceptors in human atrium: functional implicationsQ71345794
P433issue6
P921main subjectpharmacologyQ128406
P304page(s)616-628
P577publication date2004-04-30
P1433published inNaunyn-Schmiedeberg's Archives of PharmacologyQ1468251
P1476titleCloning, pharmacological characterisation and tissue distribution of a novel 5-HT4 receptor splice variant, 5-HT4(i).
P478volume369

Reverse relations

cites work (P2860)
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