Cloning and characterization of a novel human 5-HT4 receptor variant that lacks the alternatively spliced carboxy terminal exon. RT-PCR distribution in human brain and periphery of multiple 5-HT4 receptor variants

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Cloning and characterization of a novel human 5-HT4 receptor variant that lacks the alternatively spliced carboxy terminal exon. RT-PCR distribution in human brain and periphery of multiple 5-HT4 receptor variants is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/S0028-3908(01)00154-X
P698PubMed publication ID11750916

P2093author name stringPalacios JM
Mengod G
Vilaró MT
Doménech T
P2860cites workCloning, expression, and pharmacology of four human 5-hydroxytryptamine 4 receptor isoforms produced by alternative splicing in the carboxyl terminusQ24319843
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5-Hydroxytryptamine (5-HT)4 receptors in post mortem human brain tissue: distribution, pharmacology and effects of neurodegenerative diseasesQ28368154
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Inverse agonism of histamine H2 antagonist accounts for upregulation of spontaneously active histamine H2 receptorsQ28378928
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Pharmacological properties of 5-Hydroxytryptamine(4) receptor antagonists on constitutively active wild-type and mutated receptorsQ31397199
5HT4(a) and 5-HT4(b) receptors have nearly identical pharmacology and are both expressed in human atrium and ventricleQ32059490
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The 5-HT4 receptor antagonist ML10375 inhibits the constitutive activity of human 5-HT4(c) receptor.Q42132345
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Cloning, expression and pharmacology of the mouse 5-HT(4L) receptorQ42552128
The gastrointestinal prokinetic benzamide derivatives are agonists at the non-classical 5-HT receptor (5-HT4) positively coupled to adenylate cyclase in neuronsQ46224812
[3H]-GR113808 labels 5-HT4 receptors in the human and guinea-pig brain.Q46663529
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Quantitative autoradiography of 5-HT4 receptors in brains of three species using two structurally distinct radioligands, [3H]GR113808 and [3H]BIMU-1.Q46708242
5-HT4 receptors: cloning and expression of new splice variants.Q47990762
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Lesion study of the distribution of serotonin 5-HT4 receptors in rat basal ganglia and hippocampus.Q48843981
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P433issue1
P304page(s)60-73
P577publication date2002-01-01
P1433published inNeuropharmacologyQ15332439
P1476titleCloning and characterization of a novel human 5-HT4 receptor variant that lacks the alternatively spliced carboxy terminal exon. RT-PCR distribution in human brain and periphery of multiple 5-HT4 receptor variants
P478volume42

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