BPTES inhibition of hGA(124-551), a truncated form of human kidney-type glutaminase.

scientific article published on 15 October 2011

BPTES inhibition of hGA(124-551), a truncated form of human kidney-type glutaminase. is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.3109/14756366.2011.622272
P698PubMed publication ID21999665

P50authorErik W HartwickQ85097514
P2093author name stringNorman P Curthoys
P2860cites workIsolation, characterization and expression of a human brain mitochondrial glutaminase cDNAQ22253340
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Beyond aerobic glycolysis: transformed cells can engage in glutamine metabolism that exceeds the requirement for protein and nucleotide synthesisQ29617613
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Targeting mitochondrial glutaminase activity inhibits oncogenic transformationQ34807996
Glutaminase: a hot spot for regulation of cancer cell metabolism?Q37828397
Novel mechanism of inhibition of rat kidney-type glutaminase by bis-2-(5-phenylacetamido-1,2,4-thiadiazol-2-yl)ethyl sulfide (BPTES)Q39253539
Inhibition of glutaminase preferentially slows growth of glioma cells with mutant IDH1.Q39636555
Ehrlich ascites tumor cells expressing anti-sense glutaminase mRNA lose their capacity to evade the mouse immune systemQ40828562
Regulation of glutaminase activity and glutamine metabolismQ40926056
Properties of rat renal phosphate-dependent glutaminase coupled to Sepharose. Evidence that dimerization is essential for activationQ41839361
Inhibition by glutamate of phosphate-dependent glutaminase of rat kidneyQ42104953
Bacterial expression, purification, and characterization of rat kidney-type mitochondrial glutaminaseQ44578001
Phosphate-dependent glutaminase from rat kidney. Cause of increased activity in response to acidosis and identity with glutaminase from other tissuesQ53724073
P433issue6
P304page(s)861-867
P577publication date2011-10-15
P1433published inJournal of Enzyme Inhibition and Medicinal ChemistryQ15708877
P1476titleBPTES inhibition of hGA(124-551), a truncated form of human kidney-type glutaminase
P478volume27

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