and Pharmacological Activities of 14--Phenylpropyloxymorphone, a Potent Mixed Mu/Delta/Kappa-Opioid Receptor Agonist With Reduced Constipation in Mice

scientific article published on 31 August 2018

and Pharmacological Activities of 14--Phenylpropyloxymorphone, a Potent Mixed Mu/Delta/Kappa-Opioid Receptor Agonist With Reduced Constipation in Mice is …
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scholarly articleQ13442814

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P356DOI10.3389/FPHAR.2018.01002
P932PMC publication ID6127270
P698PubMed publication ID30233377

P50authorMariana SpeteaQ38545108
P2093author name stringLucia Negri
Roberta Lattanzi
Helmut Schmidhammer
Silvia Rief
P2860cites workDeltorphins: a family of naturally occurring peptides with high affinity and selectivity for delta opioid binding sitesQ24611756
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Synthesis and biological evaluation of 14-alkoxymorphinans. 18. N-substituted 14-phenylpropyloxymorphinan-6-ones with unanticipated agonist properties: extending the scope of common structure-activity relationshipsQ34191006
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Synthesis and biological evaluation of 14-alkoxymorphinans. 21. Novel 4-alkoxy and 14-phenylpropoxy derivatives of the mu opioid receptor antagonist cyprodimeQ44345593
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P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P407language of work or nameEnglishQ1860
P921main subjectpharmacologyQ128406
constipationQ178436
opioidQ427523
P304page(s)1002
P577publication date2018-08-31
P1433published inFrontiers in PharmacologyQ2681208
P1476titleIn vitro and in vivo Pharmacological Activities of 14-O-Phenylpropyloxymorphone, a Potent Mixed Mu/Delta/Kappa-Opioid Receptor Agonist With Reduced Constipation in Mice
P478volume9

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