Radiolabelled Peptides for Positron Emission Tomography and Endoradiotherapy in Oncology

scientific article published on 30 January 2020

Radiolabelled Peptides for Positron Emission Tomography and Endoradiotherapy in Oncology is …
instance of (P31):
scholarly articleQ13442814
review articleQ7318358

External links are
P356DOI10.3390/PH13020022
P932PMC publication ID7169460
P698PubMed publication ID32019275

P2093author name stringRoland Haubner
Christine Rangger
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Unexpected sensitivity of sst2 antagonists to N-terminal radiometal modificationsQ84696636
Development of Quinoline-Based Theranostic Ligands for the Targeting of Fibroblast Activation ProteinQ88295170
[68Ga]Ga-Pentixafor PET/MRI for CXCR4 Imaging of Chronic Lymphocytic Leukemia: Preliminary ResultsQ88331008
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Clinical Applications of Radiolabeled Peptides for PETQ88820027
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Targeting of the Cholecystokinin-2 Receptor with the Minigastrin Analog 177Lu-DOTA-PP-F11N: Does the Use of Protease Inhibitors Further Improve In Vivo Distribution?Q90006784
PET-Based Human Dosimetry of 68Ga-NODAGA-Exendin-4, a Tracer for β-Cell ImagingQ90100192
Development of Novel PSMA Ligands for Imaging and Therapy with Copper IsotopesQ90196809
Comparison of glucagon-like peptide-1 receptor (GLP-1R) PET/CT, SPECT/CT and 3T MRI for the localisation of occult insulinomas: evaluation of diagnostic accuracy in a prospective crossover imaging studyQ90582323
Availability of both [177Lu]Lu-DOTA-TATE and [90Y]Y-DOTATATE as PRRT agents for neuroendocrine tumors: can we evolve a rational sequential duo-PRRT protocol for large volume resistant tumors?Q90813537
Bench to Bedside: Albumin Binders for Improved Cancer Radioligand TherapiesQ90925164
Single Low-Dose Injection of Evans Blue Modified PSMA-617 Radioligand Therapy Eliminates Prostate-Specific Membrane Antigen Positive TumorsQ90935531
AAZTA5/AAZTA5-TOC: synthesis and radiochemical evaluation with 68Ga, 44Sc and 177LuQ90976884
Comparison of 68Ga-labeled RGD mono- and multimers based on a clickable siderophore-based scaffoldQ91072082
Broadening horizons with 225Ac-DOTATATE targeted alpha therapy for gastroenteropancreatic neuroendocrine tumour patients stable or refractory to 177Lu-DOTATATE PRRT: first clinical experience on the efficacy and safetyQ91211980
Intraperitoneal α-Emitting Radioimmunotherapy with 211At in Relapsed Ovarian Cancer: Long-Term Follow-up with Individual Absorbed Dose EstimationsQ91228900
Pretreatment PET/CT imaging of angiogenesis based on 18F-RGD tracer uptake may predict antiangiogenic responseQ91308795
225Ac-PSMA-617/177Lu-PSMA-617 tandem therapy of metastatic castration-resistant prostate cancer: pilot experienceQ91405943
Radiation Dosimetry and Biodistribution of 18F-PSMA-11 for PET Imaging of Prostate CancerQ91556506
An 18F-Labeled PSMA Ligand for PET/CT of Prostate Cancer: First-in-Humans Observational Study and Clinical Experience with 18F-JK-PSMA-7 During the First Year of ApplicationQ92034000
[68Ga]Ga-P16-093 as a PSMA-Targeted PET Radiopharmaceutical for Detection of Cancer: Initial Evaluation and Comparison with [68Ga]Ga-PSMA-11 in Prostate Cancer Patients Presenting with Biochemical RecurrenceQ92718603
A Systematic Review on the Role of Imaging in Early Recurrent Prostate CancerQ92726320
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68Ga-FAPI PET/CT: Tracer Uptake in 28 Different Kinds of CancerQ92898068
PSMA-Targeted Radiopharmaceuticals for Imaging and TherapyQ92943151
CXCR4-Directed Imaging in Solid TumorsQ93048437
2-(3-{1-Carboxy-5-[(6-[18F]fluoro-pyridine-3-carbonyl)-amino]-pentyl}-ureido)-pentanedioic acid, [18F]DCFPyL, a PSMA-based PET imaging agent for prostate cancerQ39449818
Strain-promoted copper-free "click" chemistry for 18F radiolabeling of bombesinQ39466193
Novel (64)Cu- and (68)Ga-labeled RGD conjugates show improved PET imaging of α(ν)β(3) integrin expression and facile radiosynthesisQ39505469
[68Ga]NODAGA-RGD for imaging αvβ3 integrin expression.Q39559499
One step radiosynthesis of 6-[(18)F]fluoronicotinic acid 2,3,5,6-tetrafluorophenyl ester ([(18)F]F-Py-TFP): a new prosthetic group for efficient labeling of biomolecules with fluorine-18.Q39750040
Clinical Translation of a Click-Labeled 18F-Octreotate Radioligand for Imaging Neuroendocrine Tumors.Q39771221
Noninvasive imaging of alphaVbeta3 function as a predictor of the antimigratory and antiproliferative effects of dasatinibQ39868638
Disparity between in vivo EGFR expression and 89Zr-labeled cetuximab uptake assessed with PET.Q39903960
A stable neurotensin-based radiopharmaceutical for targeted imaging and therapy of neurotensin receptor-positive tumoursQ39952444
Synthesis and evaluation of technetium-99m- and rhenium-labeled inhibitors of the prostate-specific membrane antigen (PSMA).Q39959750
Radiosynthesis and biodistribution of cyclic RGD peptides conjugated with novel [18F]fluorinated aldehyde-containing prosthetic groupsQ40002427
Pilot Comparison of ⁶⁸Ga-RM2 PET and ⁶⁸Ga-PSMA-11 PET in Patients with Biochemically Recurrent Prostate CancerQ40219589
Pilot prospective evaluation of (18)F-FPPRGD2 PET/CT in patients with cervical and ovarian cancerQ40270232
First (18)F-labeled tracer suitable for routine clinical imaging of sst receptor-expressing tumors using positron emission tomographyQ40550081
Use of the incretin hormone glucagon-like peptide-1 (GLP-1) for the detection of insulinomas: initial experimental resultsQ40735721
Localization of Hidden Insulinomas with ⁶⁸Ga-DOTA-Exendin-4 PET/CT: A Pilot StudyQ40913283
VPAC1 receptors for imaging breast cancer: a feasibility studyQ40991225
[177Lu]pentixather: Comprehensive Preclinical Characterization of a First CXCR4-directed Endoradiotherapeutic Agent.Q41114242
Exploring the Role of RGD-Recognizing Integrins in CancerQ41670915
89Zr-Immuno-Positron Emission Tomography in Oncology: State-of-the-Art 89Zr Radiochemistry.Q41690954
213Bi-PSMA-617 targeted alpha-radionuclide therapy in metastatic castration-resistant prostate cancer.Q41856358
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89Zr-bevacizumab PET of early antiangiogenic tumor response to treatment with HSP90 inhibitor NVP-AUY922.Q43097928
Radiohalogenated prostate-specific membrane antigen (PSMA)-based ureas as imaging agents for prostate cancerQ43193122
Direct one-step 18F-labeling of peptides via nucleophilic aromatic substitutionQ43239777
Direct labelling of peptides with 2-[18F]fluoro-2-deoxy-d-glucose ([18F]FDG).Q43295652
In vitro stability and in vivo clearance of fibrinogen or serum albumin labeled with 77Br, 131I, or 125I by direct or indirect synthetic methods.Q43500223
Noninvasive imaging of alpha(v)beta3 integrin expression using 18F-labeled RGD-containing glycopeptide and positron emission tomographyQ43561095
PET imaging of somatostatin receptors using [68GA]DOTA-D-Phe1-Tyr3-octreotide: first results in patients with meningiomasQ43662898
High-level production of alpha-particle-emitting (211)At and preparation of (211)At-labeled antibodies for clinical use.Q43755984
Pegylated Arg-Gly-Asp peptide: 64Cu labeling and PET imaging of brain tumor alphavbeta3-integrin expression.Q44275821
Cholecystokinin-B (CCK-B)/gastrin receptor targeting peptides for staging and therapy of medullary thyroid cancer and other CCK-B receptor expressing malignanciesQ44377511
Optimising conditions for radiolabelling of DOTA-peptides with 90Y, 111In and 177Lu at high specific activitiesQ44391489
Radiolabelling of isopeptide N epsilon-(gamma-glutamyl)-L-lysine by conjugation with N-succinimidyl-4-[18F]fluorobenzoateQ44523672
DOTA-NOC, a high-affinity ligand of somatostatin receptor subtypes 2, 3 and 5 for labelling with various radiometalsQ44561169
Synthesis of a New Heterobifunctional Linker, N-[4-(Aminooxy)butyl]maleimide, for Facile Access to a Thiol-Reactive 18F-Labeling AgentQ44660414
[18F]Galacto-RGD: synthesis, radiolabeling, metabolic stability, and radiation dose estimatesQ44735126
Synthesis of urea-based inhibitors as active site probes of glutamate carboxypeptidase II: efficacy as analgesic agentsQ44803462
Two-step methodology for high-yield routine radiohalogenation of peptides: (18)F-labeled RGD and octreotide analogsQ44891219
Development and characterization of clinical-grade 89Zr-trastuzumab for HER2/neu immunoPET imagingQ44944204
18F-fluorothiols: a new approach to label peptides chemoselectively as potential tracers for positron emission tomographyQ45152183
(18)F-Fluoroglucosylation of peptides, exemplified on cyclo(RGDfK).Q46059201
A series of 2-O-trifluoromethylsulfonyl-D-mannopyranosides as precursors for concomitant 18F-labeling and glycosylation by click chemistryQ46080179
microPET imaging of glioma integrin {alpha}v{beta}3 expression using (64)Cu-labeled tetrameric RGD peptideQ46115376
para-Functionalized aryl-di-tert-butylfluorosilanes as potential labeling synthons for (18)F radiopharmaceuticalsQ46155047
Biodistribution and radiation dosimetry of the integrin marker 18F-RGD-K5 determined from whole-body PET/CT in monkeys and humansQ46173308
In vivo imaging of prostate cancer using [68Ga]-labeled bombesin analog BAY86-7548.Q46234834
The biodistribution and radiation dosimetry of the Arg-Gly-Asp peptide 18F-AH111585 in healthy volunteersQ46365501
Direct procedure for the production of 211At-labeled antibodies with an epsilon-lysyl-3-(trimethylstannyl)benzamide immunoconjugateQ46429197
Development of ⁶⁸Ga-labelled DTPA galactosyl human serum albumin for liver function imagingQ46566508
Synthesis and application of [18F]FDG-maleimidehexyloxime ([18F]FDG-MHO): a [18F]FDG-based prosthetic group for the chemoselective 18F-labeling of peptides and proteinsQ46594513
Biodistribution and pharmacokinetics of the alphavbeta3-selective tracer 18F-galacto-RGD in cancer patientsQ46639250
Preparation of a promising angiogenesis PET imaging agent: 68Ga-labeled c(RGDyK)-isothiocyanatobenzyl-1,4,7-triazacyclononane-1,4,7-triacetic acid and feasibility studies in miceQ46643953
Tailored Gallium(III) chelator NOPO: synthesis, characterization, bioconjugation, and application in preclinical Ga-68-PET imaging.Q30718053
"Click labeling" with 2-[18f]fluoroethylazide for positron emission tomography.Q30831041
Radiolabeled tracers for imaging of tumor angiogenesis and evaluation of anti-angiogenic therapiesQ31059628
[(68)Ga]NODAGA-RGD - Metabolic stability, biodistribution, and dosimetry data from patients with hepatocellular carcinoma and liver cirrhosisQ31095114
64Cu-TETA-octreotide as a PET imaging agent for patients with neuroendocrine tumors.Q32053886
Imaging of integrin alpha(v)beta(3) expression in patients with malignant glioma by [18F] Galacto-RGD positron emission tomographyQ33574585
CXCR4-directed endoradiotherapy induces high response rates in extramedullary relapsed Multiple MyelomaQ33703097
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[(18)F]-NHC-BF3 adducts as water stable radio-prosthetic groups for PET imagingQ33759239
Alternative chelator for ⁸⁹Zr radiopharmaceuticals: radiolabeling and evaluation of 3,4,3-(LI-1,2-HOPO).Q33761754
Diagnostic performance of 68Ga-PSMA-11 (HBED-CC) PET/CT in patients with recurrent prostate cancer: evaluation in 1007 patientsQ33841484
In vivo transchelation of copper-64 from TETA-octreotide to superoxide dismutase in rat liver.Q33909857
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Recent progress in fluorine-18 labelled peptide radiopharmaceuticalsQ34336436
Peptidomimetics, a synthetic tool of drug discoveryQ34656152
Somatostatin analogs and radiopeptides in cancer therapyQ34972896
Pilot pharmacokinetic and dosimetric studies of (18)F-FPPRGD2: a PET radiopharmaceutical agent for imaging α(v)β(3) integrin levelsQ35062113
Radiolabeled somatostatin receptor antagonists are preferable to agonists for in vivo peptide receptor targeting of tumorsQ35103872
New Methods for Labeling RGD Peptides with Bromine-76.Q35224462
Disclosing the CXCR4 expression in lymphoproliferative diseases by targeted molecular imagingQ35227508
PET imaging of early response to the tyrosine kinase inhibitor ZD4190.Q35249646
In vivo molecular imaging of chemokine receptor CXCR4 expression in patients with advanced multiple myelomaQ35483867
Preclinical Evaluation of a Tailor-Made DOTA-Conjugated PSMA Inhibitor with Optimized Linker Moiety for Imaging and Endoradiotherapy of Prostate Cancer.Q35604902
Comparison study of [18F]FAl-NOTA-PRGD2, [18F]FPPRGD2, and [68Ga]Ga-NOTA-PRGD2 for PET imaging of U87MG tumors in miceQ35629161
Prospective Study of (68)Ga-NOTA-NFB: Radiation Dosimetry in Healthy Volunteers and First Application in Glioma PatientsQ35633357
In vitro and in vivo evaluation of a 64Cu-labeled NOTA-Bn-SCN-Aoc-bombesin analogue in gastrin-releasing peptide receptor expressing prostate cancerQ35925945
First-in-human uPAR PET: Imaging of Cancer AggressivenessQ36191589
(18)F-Alfatide II PET/CT in healthy human volunteers and patients with brain metastasesQ36225629
Synthesis and preclinical evaluation of bifunctional ligands for improved chelation chemistry of 90Y and 177Lu for targeted radioimmunotherapyQ36247600
Production of [(211)At]-astatinated radiopharmaceuticals and applications in targeted α-particle therapyQ36534262
Fluorine-18 labeling of peptides and proteins.Q36685391
In Vitro and In Vivo Comparison of Selected Ga-68 and Zr-89 Labelled Siderophores.Q36909826
First experience of 18F-alfatide in lung cancer patients using a new lyophilized kit for rapid radiofluorinationQ36931413
Gastrin-releasing Peptide Receptor Imaging in Breast Cancer Using the Receptor Antagonist (68)Ga-RM2 And PET.Q37112967
Intraperitoneal alpha-particle radioimmunotherapy of ovarian cancer patients: pharmacokinetics and dosimetry of (211)At-MX35 F(ab')2--a phase I study.Q50605886
Synthesis of [18F]RGD-K5 by catalyzed [3 + 2] cycloaddition for imaging integrin αvβ3 expression in vivo.Q50961964
Prolonged survival in secondary glioblastoma following local injection of targeted alpha therapy with 213Bi-substance P analogue.Q52715248
225Ac-PSMA-617 for PSMA-Targeted α-Radiation Therapy of Metastatic Castration-Resistant Prostate Cancer.Q52981848
Medullary thyroid carcinoma - PET/CT imaging with 68Ga-labelled gastrin and somatostatin analogues.Q52984876
First Experience with Chemokine Receptor CXCR4-Targeted PET Imaging of Patients with Solid Cancers.Q52985671
Biodistribution and radiation dosimetry of 18F-CP-18, a potential apoptosis imaging agent, as determined from PET/CT scans in healthy volunteers.Q53091381
PET imaging with a [68Ga]gallium-labelled PSMA ligand for the diagnosis of prostate cancer: biodistribution in humans and first evaluation of tumour lesions.Q53131398
Be spoilt for choice with radiolabelled RGD peptides: preclinical evaluation of ⁶⁸Ga-TRAP(RGD)₃.Q53140894
68Ga-DOTATOC versus 68Ga-DOTATATE PET/CT in functional imaging of neuroendocrine tumors.Q53192267
Synthesis and in vitro evaluation of [18F]fluoroethyl triazole labelled [Tyr3]octreotate analogues using click chemistry.Q53234108
Kit-like 18F-labeling of proteins: synthesis of 4-(di-tert-butyl[18F]fluorosilyl)benzenethiol (Si[18F]FA-SH) labeled rat serum albumin for blood pool imaging with PET.Q53375642
Positron emission tomography using [18F]Galacto-RGD identifies the level of integrin alpha(v)beta3 expression in man.Q53530857
Gluc-Lys([18F]FP)-TOCA PET in patients with SSTR-positive tumors: biodistribution and diagnostic evaluation compared with [111In]DTPA-octreotide.Q53543895
Arg-Gly-Asp constrained within cyclic pentapeptides. Strong and selective inhibitors of cell adhesion to vitronectin and laminin fragment P1.Q53686513
Small Prosthetic Groups in 18F-Radiochemistry: Useful Auxiliaries for the Design of 18F-PET Tracers.Q54246542
Site-specific stabilization of minigastrin analogs against enzymatic degradation for enhanced cholecystokinin-2 receptor targeting.Q55098217
Pharmacokinetic studies of ⁶⁸Ga-labeled Bombesin (⁶⁸Ga-BZH₃) and F-18 FDG PET in patients with recurrent gliomas and comparison to grading: preliminary results.Q55463516
First-in-human study of Lu-EB-PSMA-617 in patients with metastatic castration-resistant prostate cancerQ56523728
Automated radiosynthesis of N-succinimidyl 3-(di-tert-butyl[(18)F]fluorosilyl)benzoate ([(18)F]SiFB) for peptides and proteins radiolabeling for positron emission tomographyQ57041065
Targeted α-therapy of prostate cancer using radiolabeled PSMA inhibitors: a game changer in nuclear medicineQ57107703
Head-to-Head Comparison of 64 Cu-DOTATATE and 68 Ga-DOTATOC PET/CT: A Prospective Study of 59 Patients with Neuroendocrine TumorsQ57680025
Comparison of 68Ga-DOTATATE and 68Ga-DOTANOC PET/CT imaging in the same patient group with neuroendocrine tumoursQ57757597
Discovery of F-JK-PSMA-7, a novel PET-probe for the detection of small PSMA positive lesionsQ58617086
CXCR4-directed theranostics in oncology and inflammationQ58783862
An Overview of Targeted Alpha Therapy with Actinium and BismuthQ59796859
Development of Ac Radiopharmaceuticals: TRIUMF Perspectives and ExperiencesQ60048015
Structure and stability of hexadentate complexes of ligands based on AAZTA for efficient PET labelling with gallium-68Q60171678
Chemoselective hydrazone formation between HYNIC-functionalized peptides and 18F-fluorinated aldehydesQ60607032
[18F]galacto-RGD positron emission tomography for imaging of alphavbeta3 expression on the neovasculature in patients with squamous cell carcinoma of the head and neckQ46897615
Dual Targeting of Acute Leukemia and Supporting Niche by CXCR4-Directed Theranostics.Q47114899
Current status of theranostics in prostate cancer.Q47241139
Comparison of 68Ga-OPS202 (68Ga-NODAGA-JR11) and 68Ga-DOTATOC (68Ga-Edotreotide) PET/CT in Patients with Gastroenteropancreatic Neuroendocrine Tumors: Evaluation of Sensitivity in a Prospective Phase II Imaging StudyQ47388629
Clinical PET of neuroendocrine tumors using 64Cu-DOTATATE: first-in-humans studyQ47399002
Intra-individual comparison of 18F-PSMA-1007 and 18F-DCFPyL PET/CT in the prospective evaluation of patients with newly diagnosed prostate carcinoma: A pilot studyQ47572465
Specific inactivation of sensitized lymphocytes in vitro using antigens labelled with astatine-211Q47988801
Radiotoxicity of systemically administered 211At-labeled human/mouse chimeric monoclonal antibody: a long-term survival study with histologic analysisQ48112253
In Vivo Evaluation of ¹⁸F-SiFAlin-Modified TATE: A Potential Challenge for ⁶⁸Ga-DOTATATE, the Clinical Gold Standard for Somatostatin Receptor Imaging with PET.Q48175950
GLP-1 receptor expression in human tumors and human normal tissues: potential for in vivo targetingQ48180523
Comparison of PSMA-HBED and PSMA-I&T as diagnostic agents in prostate carcinoma.Q48188322
Imaging Characteristics and First Experience of [68Ga]THP-PSMA, a Novel Probe for Rapid Kit-Based Ga-68 Labeling and PET Imaging: Comparative Analysis with [68Ga]PSMA I&T.Q48221776
177Lu-PSMA-617 radioligand therapy in mCRPC: ready for phase III trial?Q48257941
An Eighteen-Membered Macrocyclic Ligand for Actinium-225 Targeted Alpha TherapyQ48265569
Design, synthesis, and initial evaluation of high-affinity technetium bombesin analoguesQ48487776
Automated radiosynthesis of Al[18F]PSMA-11 for large scale routine use.Q49031791
18F-AlF Labeled Peptide and Protein Conjugates as Positron Emission Tomography (PET) Imaging Pharmaceuticals.Q49797952
Targeted positron emission tomography imaging of CXCR4 expression in patients with acute myeloid leukemiaQ37140477
A practical guide to the construction of radiometallated bioconjugates for positron emission tomography.Q37172093
H(4)octapa-trastuzumab: versatile acyclic chelate system for 111In and 177Lu imaging and therapyQ37209655
(64)Cu-labeled CB-TE2A and diamsar-conjugated RGD peptide analogs for targeting angiogenesis: comparison of their biological activityQ37218456
[(64) Cu]-labelled trastuzumab: optimisation of labelling by DOTA and NODAGA conjugation and initial evaluation in miceQ37268891
Optimization of Early Response Monitoring and Prediction of Cancer Antiangiogenesis Therapy via Noninvasive PET Molecular Imaging Strategies of Multifactorial BioparametersQ37291272
Integrin α(v)β₃-targeted radiotracer (99m)Tc-3P-RGD₂ useful for noninvasive monitoring of breast tumor response to antiangiogenic linifanib therapy but not anti-integrin α(v)β₃ RGD₂ therapyQ37344824
Radiolabelled RGD peptides and peptidomimetics for tumour targetingQ37410058
Copper-64 radiopharmaceuticals for PET imaging of cancer: advances in preclinical and clinical researchQ37478003
[68Ga]Pentixafor-PET/CT for imaging of chemokine receptor CXCR4 expression in multiple myeloma - Comparison to [18F]FDG and laboratory valuesQ37541868
Comparison of the octadentate bifunctional chelator DFO*-pPhe-NCS and the clinically used hexadentate bifunctional chelator DFO-pPhe-NCS for 89Zr-immuno-PETQ37560052
68Ga-NOTA-PRGD2 PET/CT for Integrin Imaging in Patients with Lung CancerQ37575733
Glucagon-Like Peptide-1 Receptor PET/CT with 68Ga-NOTA-Exendin-4 for Detecting Localized Insulinoma: A Prospective Cohort StudyQ37581371
Peptide-based imaging agents for cancer detectionQ37585965
Longitudinal PET imaging of muscular inflammation using 18F-DPA-714 and 18F-Alfatide II and differentiation with tumorsQ37663675
Radiolabeled bombesin derivatives for preclinical oncological imaging.Q37674035
Zirconium tetraazamacrocycle complexes display extraordinary stability and provide a new strategy for zirconium-89-based radiopharmaceutical development.Q37718007
(2S)-2-(3-(1-Carboxy-5-(4-211At-Astatobenzamido)Pentyl)Ureido)-Pentanedioic Acid for PSMA-Targeted α-Particle Radiopharmaceutical TherapyQ37722429
Homeostatic chemokine receptors and organ-specific metastasisQ37922092
Radiobromine-labelled tracers for positron emission tomography: possibilities and pitfalls.Q37970739
PET tracers based on Zirconium-89.Q37970745
Actinium-225 in targeted alpha-particle therapeutic applications.Q37971807
A review on CXCR4/CXCL12 axis in oncology: no place to hide.Q38017493
Click-to-Chelate: development of technetium and rhenium-tricarbonyl labeled radiopharmaceuticalsQ38088564
Matching chelators to radiometals for radiopharmaceuticalsQ38156660
Chelators for copper radionuclides in positron emission tomography radiopharmaceuticalsQ38172069
PET radiopharmaceuticals for imaging integrin expression: tracers in clinical studies and recent developments.Q38228356
GLP-1 and exendin-4 for imaging endocrine pancreas. A review. Labelled glucagon-like peptide-1 analogues: past, present and futureQ38365438
Molecular Pathways: Targeting the CXCR4-CXCL12 Axis--Untapped Potential in the Tumor MicroenvironmentQ38551844
Preclinical Evaluation of 18F-PSMA-1007, a New Prostate-Specific Membrane Antigen Ligand for Prostate Cancer Imaging.Q38735685
Theranostic Perspectives in Prostate Cancer with the Gastrin-Releasing Peptide Receptor Antagonist NeoBOMB1: Preclinical and First Clinical ResultsQ38753711
Toward the Optimization of Bombesin-Based Radiotracers for Tumor Targeting.Q38780032
PSA-Stratified Performance of 18F- and 68Ga-PSMA PET in Patients with Biochemical Recurrence of Prostate Cancer.Q38788408
Preclinical and first clinical experience with the gastrin-releasing peptide receptor-antagonist [⁶⁸Ga]SB3 and PET/CT.Q38814811
Comparison of the Therapeutic Response to Treatment with a 177Lu-Labeled Somatostatin Receptor Agonist and Antagonist in Preclinical Models.Q38823932
P275copyright licenseCreative Commons Attribution 4.0 InternationalQ20007257
P6216copyright statuscopyrightedQ50423863
P433issue2
P921main subjectpositron emission tomographyQ208376
P577publication date2020-01-30
P1433published inPharmaceuticalsQ15750667
P1476titleRadiolabelled Peptides for Positron Emission Tomography and Endoradiotherapy in Oncology
P478volume13

Reverse relations

Q97588200Identification of a suitable peptidic molecular platform for the development of NPY(Y1)R-specific imaging agentscites workP2860