scholarly article | Q13442814 |
P356 | DOI | 10.1002/CMDC.201900170 |
P698 | PubMed publication ID | 30957949 |
P50 | author | Klaus Theodor Wanner | Q87805156 |
P2093 | author name string | Georg Höfner | |
Maren Schaarschmidt | |||
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Deletion of the betaine-GABA transporter (BGT1; slc6a12) gene does not affect seizure thresholds of adult mice | Q34175243 | ||
The betaine-GABA transporter (BGT1, slc6a12) is predominantly expressed in the liver and at lower levels in the kidneys and at the brain surface. | Q34231212 | ||
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Different Binding Modes of Small and Large Binders of GAT1. | Q40068020 | ||
Stereoselective central nervous system effects of the R- and S-isomers of the GABA uptake blocker N-(4, 4-di-(3-methylthien-2-yl)but-3-enyl) nipecotic acid in the rat. | Q41977092 | ||
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Tiagabine and gabapentin for the management of chronic pain | Q46542324 | ||
Synthesis of Allene Substituted Nipecotic Acids by Allenylation of Terminal Alkynes. | Q48140476 | ||
Atroposelective Synthesis of Axially Chiral Biaryls by Palladium-Catalyzed Asymmetric C-H Olefination Enabled by a Transient Chiral Auxiliary | Q48192962 | ||
Synthesis of 4-substituted nipecotic acid derivatives and their evaluation as potential GABA uptake inhibitors. | Q50864675 | ||
Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives with N-Arylalkynyl Substituents. | Q51167808 | ||
Atroposelective Synthesis of Axially Chiral Biaryls by Palladium-Catalyzed Asymmetric C−H Olefination Enabled by a Transient Chiral Auxiliary | Q59755116 | ||
MS-binding assays: kinetic, saturation, and competitive experiments based on quantitation of bound marker as exemplified by the GABA transporter mGAT1 | Q80067141 | ||
Mild-condition synthesis of allenes from alkynes and aldehydes mediated by tetrahydroisoquinoline (THIQ) | Q86830004 | ||
Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions | Q86938754 | ||
P433 | issue | 12 | |
P304 | page(s) | 1135-1151 | |
P577 | publication date | 2019-05-08 | |
P1433 | published in | ChemMedChem | Q2962252 |
P1476 | title | Synthesis and Biological Evaluation of Nipecotic Acid and Guvacine Derived 1,3-Disubstituted Allenes as Inhibitors of Murine GABA Transporter mGAT1 | |
P478 | volume | 14 |
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