Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions

scientific article published on 18 December 2015

Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1002/CMDC.201500490
P698PubMed publication ID26683881

P50authorJörg PabelQ73375603
Klaus Theodor WannerQ87805156
P2093author name stringMarilena Petrera
Georg Höfner
Lars Allmendinger
Thomas Wein
Miriam Sindelar
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P433issue5
P304page(s)519-538
P577publication date2015-12-18
P1433published inChemMedChemQ2962252
P1476titleDevelopment of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives by Suzuki-Miyaura Cross-Coupling Reactions
P478volume11

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cites work (P2860)
Q51167808Development of Highly Potent GAT1 Inhibitors: Synthesis of Nipecotic Acid Derivatives with N-Arylalkynyl Substituents.
Q48144959Development of Non-GAT1-Selective Inhibitors: Challenges and Achievements
Q61805435GRID-independent molecular descriptor analysis and molecular docking studies to mimic the binding hypothesis of γ-aminobutyric acid transporter 1 (GAT1) inhibitors
Q90431734N-Substituted Nipecotic Acids as (S)-SNAP-5114 Analogues with Modified Lipophilic Domains
Q92921913Synthesis and Biological Evaluation of Nipecotic Acid and Guvacine Derived 1,3-Disubstituted Allenes as Inhibitors of Murine GABA Transporter mGAT1

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