Selective N-Hydroxyhydantoin Carbamate Inhibitors of Mammalian Serine Hydrolases

scientific article published on 25 June 2015

Selective N-Hydroxyhydantoin Carbamate Inhibitors of Mammalian Serine Hydrolases is …
instance of (P31):
scholarly articleQ13442814

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P356DOI10.1016/J.CHEMBIOL.2015.05.018
P932PMC publication ID4527528
P698PubMed publication ID26120000
P5875ResearchGate publication ID279457867

P50authorBenjamin CravattQ4888433
Hyeon-Cheol LeeQ57334431
Armand B CognettaQ61456374
P2093author name stringMicah J Niphakis
Jonathan J Hulce
Michael L Martini
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Dual inhibition of alpha/beta-hydrolase domain 6 and fatty acid amide hydrolase increases endocannabinoid levels in neurons.Q35309312
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The first wave: HCV NS3 protease inhibitors telaprevir and boceprevirQ38063182
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A potent and selective inhibitor of KIAA1363/AADACL1 that impairs prostate cancer pathogenesisQ39554498
Palmitoyl:protein thioesterase (PPT1) inhibitors can act as pharmacological chaperones in infantile Batten diseaseQ39722105
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Endocannabinoid biosynthesis proceeding through glycerophospho-N-acyl ethanolamine and a role for alpha/beta-hydrolase 4 in this pathwayQ41791622
Direct visualization of serine hydrolase activities in complex proteomes using fluorescent active site-directed probesQ43979860
A functional proteomic strategy to discover inhibitors for uncharacterized hydrolasesQ46044614
The antiproliferative agent didemnin B uncompetitively inhibits palmitoyl protein thioesteraseQ47813181
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Beta-lactams as selective chemical probes for the in vivo labeling of bacterial enzymes involved in cell wall biosynthesis, antibiotic resistance, and virulence.Q50777469
Functional and quantitative proteomics using SILACQ57369727
Purification of rabbit myocardial cytosolic acyl-CoA hydrolase, identity with lysophospholipase, and modulation of enzymic activity by endogenous cardiac amphiphilesQ72568603
A rapid fluorogenic palmitoyl-protein thioesterase assay: pre- and postnatal diagnosis of INCLQ77223127
P4510describes a project that usesImageJQ1659584
P433issue7
P304page(s)928-937
P577publication date2015-06-25
P1433published inChemistry and BiologyQ15758410
P1476titleSelective N-Hydroxyhydantoin Carbamate Inhibitors of Mammalian Serine Hydrolases
P478volume22

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Q47266601"Inverse Drug Discovery" Strategy To Identify Proteins That Are Targeted by Latent Electrophiles As Exemplified by Aryl Fluorosulfates
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