Highly Constrained Bicyclic Scaffolds for the Discovery of Protease-Stable Peptides via mRNA Display

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Highly Constrained Bicyclic Scaffolds for the Discovery of Protease-Stable Peptides via mRNA Display is …
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scholarly articleQ13442814

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P356DOI10.1021/ACSCHEMBIO.6B01006
P932PMC publication ID5443354
P698PubMed publication ID28146347

P50authorEmil S IqbalQ64181851
Matthew C T HartmanQ89232649
Teresa M. PrzytyckaQ37371892
P2093author name stringJan Hoinka
David E Hacker
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Integrin-Targeting Knottin Peptide-Drug Conjugates Are Potent Inhibitors of Tumor Cell Proliferation.Q48199301
Quantitative comparison of the relative cell permeability of cyclic and linear peptidesQ53545017
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Rapid and quantitative cyclization of multiple peptide loops onto synthetic scaffolds for structural mimicry of protein surfacesQ81617617
Improved proteolytic stability of chicken cathelicidin-2 derived peptides by D-amino acid substitutions and cyclizationQ83534410
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Ribosomal Synthesis of Natural-Product-Like Bicyclic Peptides in Escherichia coliQ36070579
Analysis and optimization of copper-catalyzed azide-alkyne cycloaddition for bioconjugationQ36136380
Screening of cyclic peptide phage libraries identifies ligands that bind streptavidin with high affinitiesQ36671737
Identification of avidin and streptavidin binding motifs among peptides selected from a synthetic peptide library consisting solely of D‐amino acidsQ36871020
Engineered knottin peptide enables noninvasive optical imaging of intracranial medulloblastomaQ37157248
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Cell-permeable bicyclic peptide inhibitors against intracellular proteinsQ38980364
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P433issue3
P304page(s)795-804
P577publication date2017-02-01
P1433published inACS Chemical BiologyQ165583
P1476titleHighly Constrained Bicyclic Scaffolds for the Discovery of Protease-Stable Peptides via mRNA Display
P478volume12

Reverse relations

cites work (P2860)
Q52669426An anti-PDGFRβ aptamer for selective delivery of small therapeutic peptide to cardiac cells.
Q36394825Bicyclic Peptides as Next-Generation Therapeutics.
Q88524917Cyclization of peptides with two chemical bridges affords large scaffold diversities
Q47765958Directed Evolution of Glycopeptides Using mRNA Display
Q61795450Discovery of Nonstandard Macrocyclic Peptides as Noncompetitive Inhibitors of the Zika Virus NS2B-NS3 Protease
Q48171005Ribosomal incorporation of backbone modified amino acids via an editing-deficient aminoacyl-tRNA synthetase
Q61814870Toxin Neutralization Using Alternative Binding Proteins

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