Regulation of Estrogen Receptor α by the SET7 Lysine Methyltransferase

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Regulation of Estrogen Receptor α by the SET7 Lysine Methyltransferase is …
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scholarly articleQ13442814

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P356DOI10.1016/J.MOLCEL.2008.03.022
P3181OpenCitations bibliographic resource ID948904
P932PMC publication ID2567917
P698PubMed publication ID18471979
P5875ResearchGate publication ID5379563

P2093author name stringXiaodong Cheng
Junmin Peng
Da Jia
Robert E Collins
Doris R Powell
Paula M Vertino
Dipali Sharma
Krithika Subramanian
Priya Kapoor-Vazirani
P2860cites workRegulation of chromatin structure by site-specific histone H3 methyltransferasesQ24290115
p53 is regulated by the lysine demethylase LSD1Q24292925
Structural basis for the methylation site specificity of SET7/9Q24301341
Regulation of p53 activity through lysine methylationQ24311514
LSD1 demethylates repressive histone marks to promote androgen-receptor-dependent transcriptionQ24312958
Repression of p53 activity by Smyd2-mediated methylationQ24315991
Identification of the MLL2 complex as a coactivator for estrogen receptor alphaQ24316007
Gene-specific modulation of TAF10 function by SET9-mediated methylationQ24337399
Regulation of coactivator complex assembly and function by protein arginine methylation and demethyliminationQ24556492
In vitro and in vivo analyses of a Phe/Tyr switch controlling product specificity of histone lysine methyltransferasesQ24645737
Structural basis for the product specificity of histone lysine methyltransferasesQ24646957
Set9, a novel histone H3 methyltransferase that facilitates transcription by precluding histone tail modifications required for heterochromatin formationQ24672514
The estrogen receptor-alpha A908G (K303R) mutation occurs at a low frequency in invasive breast tumors: results from a population-based studyQ25257794
TMS1, a novel proapoptotic caspase recruitment domain protein, is a target of methylation-induced gene silencing in human breast cancersQ28139273
NSD1 is essential for early post-implantation development and has a catalytically active SET domainQ28593118
Dynamic Regulation of Histone Lysine Methylation by DemethylasesQ29036779
Methylation of lysine 4 on histone H3: intricacy of writing and reading a single epigenetic markQ29614516
Genome-wide analysis of estrogen receptor binding sitesQ29614765
Cellular and molecular pharmacology of antiestrogen action and resistanceQ31921111
Oestrogen receptors - an overviewQ33711233
The SRC family of nuclear receptor coactivatorsQ33860695
Synergistic enhancement of nuclear receptor function by p160 coactivators and two coactivators with protein methyltransferase activitiesQ33922863
Direct acetylation of the estrogen receptor alpha hinge region by p300 regulates transactivation and hormone sensitivityQ33940612
Purification and functional characterization of a histone H3-lysine 4-specific methyltransferase.Q34108153
Nuclear receptor coregulators: multiple modes of modificationQ34537625
Ligand-dependent transcription of estrogen receptor alpha is mediated by the ubiquitin ligase EFP.Q34617201
Acetylation of estrogen receptor alpha by p300 at lysines 266 and 268 enhances the deoxyribonucleic acid binding and transactivation activities of the receptorQ34698474
Nuclear receptor modifications and endocrine cell proliferationQ35207718
Histone H3 lysine 9 methyltransferase G9a is a transcriptional coactivator for nuclear receptorsQ35589266
Estrogen receptor alpha is a putative substrate for the BRCA1 ubiquitin ligaseQ35749504
Association between the estrogen receptor alpha A908G mutation and outcomes in invasive breast cancerQ35794355
Risk factors for breast cancer characterized by the estrogen receptor alpha A908G (K303R) mutationQ35906333
Effect of tamoxifen on Ki67 labelling index in human breast tumours and its relationship to oestrogen and progesterone receptor status.Q35976106
Histone methylation-dependent mechanisms impose ligand dependency for gene activation by nuclear receptorsQ36014589
Effects of endocrine therapy on steroid-receptor content of breast cancerQ36046259
Coregulators in nuclear estrogen receptor action: from concept to therapeutic targetingQ36361043
A histone methyltransferase is required for maximal response to female sex hormonesQ36701489
Proteasome-dependent degradation of the human estrogen receptorQ37160826
Lysine trimethylation of retinoic acid receptor-alpha: a novel means to regulate receptor functionQ38305996
An assessment of the role of domain F and PEST sequences in estrogen receptor half-life and bioactivityQ38313711
Tamoxifen resistance by a conformational arrest of the estrogen receptor alpha after PKA activation in breast cancerQ38340180
Cyclic, proteasome-mediated turnover of unliganded and liganded ERalpha on responsive promoters is an integral feature of estrogen signalingQ38356127
Differential regulation of estrogen receptor alpha turnover and transactivation by Mdm2 and stress-inducing agentsQ40124566
P21-activated kinase 1 regulation of estrogen receptor-alpha activation involves serine 305 activation linked with serine 118 phosphorylationQ40321973
E6AP and calmodulin reciprocally regulate estrogen receptor stability.Q40346484
Phosphorylation of estrogen receptor alpha blocks its acetylation and regulates estrogen sensitivity.Q40479849
Ligand-dependent switching of ubiquitin-proteasome pathways for estrogen receptorQ40493369
Neurite-localized estrogen receptor-alpha mediates rapid signaling by estrogenQ40634138
Proteasome-mediated proteolysis of estrogen receptor: a novel component in autologous down-regulationQ40930380
Calmodulin is a selective modulator of estrogen receptorsQ43974253
Ubiquitination of the Rat Uterine Estrogen Receptor: Dependence on EstradiolQ71970742
A hypersensitive estrogen receptor-alpha mutation in premalignant breast lesionsQ74181062
The human estrogen receptor-alpha is a ubiquitinated protein whose stability is affected differentially by agonists, antagonists, and selective estrogen receptor modulatorsQ74265958
It takes a PHD to interpret histone methylationQ79853386
P433issue3
P407language of work or nameEnglishQ1860
P921main subjectcell biologyQ7141
estrogenQ277954
P304page(s)336-47
P577publication date2008-05-09
P1433published inMolecular CellQ3319468
P1476titleRegulation of Estrogen Receptor α by the SET7 Lysine Methyltransferase
P478volume30

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